Trial Outcomes & Findings for Efficacy of an Intranasal Testosterone Product (NCT NCT01252745)

NCT ID: NCT01252745

Last Updated: 2018-05-23

Results Overview

Recruitment status

COMPLETED

Study phase

PHASE2

Target enrollment

22 participants

Primary outcome timeframe

24 hours

Results posted on

2018-05-23

Participant Flow

Participant milestones

Participant milestones
Measure
10.0 mg Testosterone t.i.d.
TBS-1 syringes pre-filled with 125 μL 4.0% gel to deliver 5.0 mg of Testosterone per nostril (intra-nasal) given t.i.d. at 2100, 0700, and 1300 hours. (total dose 30 mg/day)
13.5 mg Testosterone b.i.d.
TBS-1 syringes pre-filled with 150 μL 4.5% gel to deliver 6.75 mg of Testosterone per nostril (intra-nasal) given b.i.d. at 2100 and 0700 hours. (total dose 27.0 mg/day)
11.25 mg Testosterone t.i.d.
TBS-1 syringes pre-filled with 125 μL 4.5% gel to deliver 5.625 mg of Testosterone per nostril (intra-nasal) given t.i.d. at 2100, 0700, and 1300 hours. (total dose 33.75 mg/day)
Overall Study
STARTED
8
7
7
Overall Study
COMPLETED
8
7
7
Overall Study
NOT COMPLETED
0
0
0

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

Efficacy of an Intranasal Testosterone Product

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
10.0 mg Testosterone t.i.d.
n=8 Participants
TBS-1 syringes pre-filled with 125 μL 4.0% gel to deliver 5.0 mg of Testosterone per nostril (intra-nasal) given t.i.d. at 2100, 0700, and 1300 hours. (total dose 30 mg/day)
13.5 mg Testosterone b.i.d.
n=7 Participants
TBS-1 syringes pre-filled with 150 μL 4.5% gel to deliver 6.75 mg of Testosterone per nostril (intra-nasal) given b.i.d. at 2100 and 0700 hours. (total dose 27.0 mg/day)
11.25 mg Testosterone t.i.d.
n=7 Participants
TBS-1 syringes pre-filled with 125 μL 4.5% gel to deliver 5.625 mg of Testosterone per nostril (intra-nasal) given t.i.d. at 2100, 0700, and 1300 hours. (total dose 33.75 mg/day)
Total
n=22 Participants
Total of all reporting groups
Age, Continuous
52.38 years
STANDARD_DEVIATION 12.55 • n=93 Participants
53.86 years
STANDARD_DEVIATION 11.04 • n=4 Participants
51.57 years
STANDARD_DEVIATION 9.90 • n=27 Participants
52.59 years
STANDARD_DEVIATION 10.78 • n=483 Participants
Sex: Female, Male
Female
0 Participants
n=93 Participants
0 Participants
n=4 Participants
0 Participants
n=27 Participants
0 Participants
n=483 Participants
Sex: Female, Male
Male
8 Participants
n=93 Participants
7 Participants
n=4 Participants
7 Participants
n=27 Participants
22 Participants
n=483 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
4 Participants
n=93 Participants
3 Participants
n=4 Participants
3 Participants
n=27 Participants
10 Participants
n=483 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
4 Participants
n=93 Participants
4 Participants
n=4 Participants
4 Participants
n=27 Participants
12 Participants
n=483 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
0 Participants
n=93 Participants
0 Participants
n=4 Participants
0 Participants
n=27 Participants
0 Participants
n=483 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=93 Participants
0 Participants
n=4 Participants
0 Participants
n=27 Participants
0 Participants
n=483 Participants
Race (NIH/OMB)
Asian
0 Participants
n=93 Participants
0 Participants
n=4 Participants
0 Participants
n=27 Participants
0 Participants
n=483 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=93 Participants
0 Participants
n=4 Participants
0 Participants
n=27 Participants
0 Participants
n=483 Participants
Race (NIH/OMB)
Black or African American
0 Participants
n=93 Participants
0 Participants
n=4 Participants
1 Participants
n=27 Participants
1 Participants
n=483 Participants
Race (NIH/OMB)
White
8 Participants
n=93 Participants
7 Participants
n=4 Participants
6 Participants
n=27 Participants
21 Participants
n=483 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=93 Participants
0 Participants
n=4 Participants
0 Participants
n=27 Participants
0 Participants
n=483 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=93 Participants
0 Participants
n=4 Participants
0 Participants
n=27 Participants
0 Participants
n=483 Participants
Region of Enrollment
United States
8 Participants
n=93 Participants
7 Participants
n=4 Participants
7 Participants
n=27 Participants
22 Participants
n=483 Participants

PRIMARY outcome

Timeframe: 24 hours

Outcome measures

Outcome measures
Measure
10.0 mg Testosterone t.i.d.
n=8 Participants
TBS-1 syringes pre-filled with 125 μL 4.0% gel to deliver 5.0 mg of Testosterone per nostril (intra-nasal) given t.i.d. at 2100, 0700, and 1300 hours. (total dose 30 mg/day)
13.5 mg Testosterone b.i.d.
n=7 Participants
TBS-1 syringes pre-filled with 150 μL 4.5% gel to deliver 6.75 mg of Testosterone per nostril (intra-nasal) given b.i.d. at 2100 and 0700 hours. (total dose 27.0 mg/day)
11.25 mg Testosterone t.i.d.
n=7 Participants
TBS-1 syringes pre-filled with 125 μL 4.5% gel to deliver 5.625 mg of Testosterone per nostril (intra-nasal) given t.i.d. at 2100, 0700, and 1300 hours. (total dose 33.75 mg/day)
Cmax of Serum Testosterone
830 ng/dL
Standard Deviation 188
1050 ng/dL
Standard Deviation 463
883 ng/dL
Standard Deviation 346

PRIMARY outcome

Timeframe: 24 hours

Outcome measures

Outcome measures
Measure
10.0 mg Testosterone t.i.d.
n=8 Participants
TBS-1 syringes pre-filled with 125 μL 4.0% gel to deliver 5.0 mg of Testosterone per nostril (intra-nasal) given t.i.d. at 2100, 0700, and 1300 hours. (total dose 30 mg/day)
13.5 mg Testosterone b.i.d.
n=7 Participants
TBS-1 syringes pre-filled with 150 μL 4.5% gel to deliver 6.75 mg of Testosterone per nostril (intra-nasal) given b.i.d. at 2100 and 0700 hours. (total dose 27.0 mg/day)
11.25 mg Testosterone t.i.d.
n=7 Participants
TBS-1 syringes pre-filled with 125 μL 4.5% gel to deliver 5.625 mg of Testosterone per nostril (intra-nasal) given t.i.d. at 2100, 0700, and 1300 hours. (total dose 33.75 mg/day)
Cavg of Serum Testosterone
413 ng/dL
Standard Deviation 138
408 ng/dL
Standard Deviation 147
396 ng/dL
Standard Deviation 110

PRIMARY outcome

Timeframe: 24 hours

Outcome measures

Outcome measures
Measure
10.0 mg Testosterone t.i.d.
n=8 Participants
TBS-1 syringes pre-filled with 125 μL 4.0% gel to deliver 5.0 mg of Testosterone per nostril (intra-nasal) given t.i.d. at 2100, 0700, and 1300 hours. (total dose 30 mg/day)
13.5 mg Testosterone b.i.d.
n=7 Participants
TBS-1 syringes pre-filled with 150 μL 4.5% gel to deliver 6.75 mg of Testosterone per nostril (intra-nasal) given b.i.d. at 2100 and 0700 hours. (total dose 27.0 mg/day)
11.25 mg Testosterone t.i.d.
n=7 Participants
TBS-1 syringes pre-filled with 125 μL 4.5% gel to deliver 5.625 mg of Testosterone per nostril (intra-nasal) given t.i.d. at 2100, 0700, and 1300 hours. (total dose 33.75 mg/day)
AUC0-t of Serum Testosterone
9920.07 ng.h/dL
Standard Deviation 3300.65
9781.39 ng.h/dL
Standard Deviation 3532.43
9505.03 ng.h/dL
Standard Deviation 2650.59

Adverse Events

10.0 mg Testosterone t.i.d.

Serious events: 0 serious events
Other events: 4 other events
Deaths: 0 deaths

13.5 mg Testosterone b.i.d.

Serious events: 0 serious events
Other events: 2 other events
Deaths: 0 deaths

11.25 mg Testosterone t.i.d.

Serious events: 0 serious events
Other events: 0 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
10.0 mg Testosterone t.i.d.
n=8 participants at risk
TBS-1 syringes pre-filled with 125 μL 4.0% gel to deliver 5.0 mg of Testosterone per nostril (intra-nasal) given t.i.d. at 2100, 0700, and 1300 hours. (total dose 30 mg/day)
13.5 mg Testosterone b.i.d.
n=7 participants at risk
TBS-1 syringes pre-filled with 150 μL 4.5% gel to deliver 6.75 mg of Testosterone per nostril (intra-nasal) given b.i.d. at 2100 and 0700 hours. (total dose 27.0 mg/day)
11.25 mg Testosterone t.i.d.
n=7 participants at risk
TBS-1 syringes pre-filled with 125 μL 4.5% gel to deliver 5.625 mg of Testosterone per nostril (intra-nasal) given t.i.d. at 2100, 0700, and 1300 hours. (total dose 33.75 mg/day)
Nervous system disorders
Dizziness
25.0%
2/8 • Number of events 2 • 1 month
0.00%
0/7 • 1 month
0.00%
0/7 • 1 month
Skin and subcutaneous tissue disorders
Pain of skin
12.5%
1/8 • Number of events 1 • 1 month
0.00%
0/7 • 1 month
0.00%
0/7 • 1 month
Skin and subcutaneous tissue disorders
Excoriation
12.5%
1/8 • Number of events 1 • 1 month
0.00%
0/7 • 1 month
0.00%
0/7 • 1 month
Respiratory, thoracic and mediastinal disorders
Respiratory tract congestion
0.00%
0/8 • 1 month
14.3%
1/7 • Number of events 1 • 1 month
0.00%
0/7 • 1 month
Gastrointestinal disorders
Gastrooesophageal reflux disease
0.00%
0/8 • 1 month
14.3%
1/7 • Number of events 1 • 1 month
0.00%
0/7 • 1 month
Blood and lymphatic system disorders
Anemia
12.5%
1/8 • Number of events 1 • 1 month
0.00%
0/7 • 1 month
0.00%
0/7 • 1 month

Additional Information

Vice President

Acerus Pharmaceuticals Corporation

Phone: (416) 679-0776

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place

Restriction type: GT60