Investigation of Efficacy, Safety and Tolerability of Once and Twice Daily Doses of AZD1981 in Asthmatic Patients

NCT ID: NCT01197794

Last Updated: 2013-11-06

Study Results

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

1144 participants

Study Classification

INTERVENTIONAL

Study Start Date

2010-10-31

Study Completion Date

2012-02-29

Brief Summary

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The study will assess the efficacy, safety and tolerability of AZD1981 compared to non-active compound in asthmatic patients.

Detailed Description

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Conditions

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Asthma Patients

Keywords

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Efficacy safety tolerability dose finding asthma patients

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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AZD1981 10 mg

AZD1981 10 mg

Group Type EXPERIMENTAL

AZD1981

Intervention Type DRUG

AZD1981 twice daily

AZD1981 40 mg

AZD1981 40 mg

Group Type EXPERIMENTAL

AZD1981

Intervention Type DRUG

AZD1981 twice daily

AZD1981 100 mg

AZD1981 100 mg

Group Type EXPERIMENTAL

AZD1981

Intervention Type DRUG

AZD1981 twice daily

AZD1981 400 mg

AZD1981 400 mg

Group Type EXPERIMENTAL

AZD1981

Intervention Type DRUG

AZD1981 twice daily

AZD1981 80 mg

AZD1981 80 mg

Group Type EXPERIMENTAL

AZD1981

Intervention Type DRUG

AZD1981 once daily

AZD1981 200 mg

AZD1981 200 mg

Group Type EXPERIMENTAL

AZD1981

Intervention Type DRUG

AZD1981 once daily

Placebo

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Placebo to match AZD1981

Interventions

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AZD1981

AZD1981 twice daily

Intervention Type DRUG

AZD1981

AZD1981 once daily

Intervention Type DRUG

Placebo

Placebo to match AZD1981

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Men and women. Women must be surgically sterilized/postmenopausal or use double barrier method contraception
* 6 months history of asthma according to ATS definition
* Prescribed daily dose of ICS and LABA for at least 3 months prior to Visit 2
* Pre-bronchodilator FEV1 of 40 to 85 % of predicted normal
* A total ACQ5 score of 1.5 or more

Exclusion Criteria

* Respiratory infection significantly affecting the asthma
* Any significant disease and disorder that may put the patient at risk or influence study results
* Any clinically relevant abnormal findings
* A smoking history of more than 10 pack years
* Intake of oral, rectal or parenteral glucocorticosteroids
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Chris O'Brien, MD

Role: STUDY_DIRECTOR

AstraZeneca

Locations

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Research Site

Fullerton, California, United States

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Los Angeles, California, United States

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Mission Viejo, California, United States

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Rolling Hills Estates, California, United States

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San Diego, California, United States

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San Jose, California, United States

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Wheaton, Maryland, United States

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North Dartmouth, Massachusetts, United States

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Bellevue, Nebraska, United States

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Sylvania, Ohio, United States

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Oklahoma City, Oklahoma, United States

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Medford, Oregon, United States

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Portland, Oregon, United States

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Collegeville, Pennsylvania, United States

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Pittsburgh, Pennsylvania, United States

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Charleston, South Carolina, United States

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Clinton, South Carolina, United States

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Waco, Texas, United States

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Tacoma, Washington, United States

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Buenos Aires, Argentina, Argentina

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Quilmes, Buenos Aires, Argentina

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Mendoza, Mendoza Province, Argentina

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Rosario, Santa Fe Province, Argentina

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San Miguel de Tucumán, Tucumán Province, Argentina

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Porto Alegre, Brasil, Brazil

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Vitória, Espírito Santo, Brazil

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Belo Horizonte, Minas Gerais, Brazil

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Juiz de Fora, Minas Gerais, Brazil

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Porto Alegre, Rio Grande do Sul, Brazil

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Florian Polis, Santa Catarina, Brazil

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Santo André, São Paulo, Brazil

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São Paulo, São Paulo, Brazil

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Yanagawa, Fukuoka, Japan

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Hiroshima, Hiroshima, Japan

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Asahikawa, Hokkaido, Japan

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Chitose, Hokkaido, Japan

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Kitahiroshima, Hokkaido, Japan

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Obihiro, Hokkaido, Japan

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Sapporo, Hokkaido, Japan

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Tomakomai, Hokkaido, Japan

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Himeji, Hyōgo, Japan

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Naka-gun, Ibaraki, Japan

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Sakaidechō, Kagawa-ken, Japan

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Fujisawa-shi, Kanagawa, Japan

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Yokohama, Kanagawa, Japan

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Kochi, Kochi, Japan

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Kyoto, Kyoto, Japan

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Nagaoka, Niigata, Japan

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Beppu, Oita Prefecture, Japan

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Ōita, Oita Prefecture, Japan

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Kurashiki-shi, Okayama-ken, Japan

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Matsue, Shimane, Japan

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Chuo-ku, Tokyo, Japan

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Chūō, Tokyo, Japan

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Itabashi-ku, Tokyo, Japan

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Kodaira, Tokyo, Japan

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Nakano-ku, Tokyo, Japan

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Ohota-ku, Tokyo, Japan

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México, D.f., Mexico

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Tijuana, Estado de Baja California, Mexico

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Morelia, Michoacán, Mexico

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Monterrey, Nuevo León, Mexico

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Guadalajara, , Mexico

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Constanța, Constanța County, Romania

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Brasov, , Romania

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Bucharest, , Romania

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Cluj-Napoca, , Romania

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Iași, , Romania

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Tg. Mures, , Romania

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Moscow, Russia, Russia

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Yekaterinburg, Russia, Russia

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Novosibirsk, , Russia

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Saint Petersburg, , Russia

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Vladikavkaz, , Russia

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Banská Bystrica, , Slovakia

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Bardejov, , Slovakia

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Bratislava, , Slovakia

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Dunajská Streda, , Slovakia

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Hnúšťa, , Slovakia

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Komárno, , Slovakia

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Košice, , Slovakia

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Levice, , Slovakia

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Liptovský Hrádok, , Slovakia

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Liptovský Mikuláš, , Slovakia

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Prešov, , Slovakia

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Rimavská Sobota, , Slovakia

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Ružomberok, , Slovakia

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Trenčín, , Slovakia

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Zvolen, , Slovakia

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Lyttleton, Centurion, South Africa

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Durban, KwaZulu-Natal, South Africa

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Cape Town, South Africa, South Africa

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Durban, South Africa, South Africa

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eMkhomazi, South Africa, South Africa

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Durbanville, , South Africa

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eManzimtoti, , South Africa

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Pretoria, , South Africa

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Dnipropetrovsk, , Ukraine

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Donetsk, , Ukraine

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Kharkiv, , Ukraine

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Kyiv, , Ukraine

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Odesa, , Ukraine

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Poltava, , Ukraine

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Vinytsa, , Ukraine

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Zaporizhzhya, , Ukraine

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Countries

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United States Argentina Brazil Japan Mexico Romania Russia Slovakia South Africa Ukraine

References

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Bateman ED, O'Brien C, Rugman P, Luke S, Ivanov S, Uddin M. Efficacy and safety of the CRTh2 antagonist AZD1981 as add-on therapy to inhaled corticosteroids and long-acting beta2-agonists in patients with atopic asthma. Drug Des Devel Ther. 2018 May 4;12:1093-1106. doi: 10.2147/DDDT.S147389. eCollection 2018.

Reference Type DERIVED
PMID: 29765200 (View on PubMed)

Other Identifiers

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2010-020407-73

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

D9830C00008

Identifier Type: -

Identifier Source: org_study_id