Safety and Tolerability Study of GSK1120212, a MEK Inhibitor, in Combination With Docetaxel, Erlotinib, Pemetrexed, Pemetrexed + Carboplatin, Pemetrexed + Cisplatin, or Nab-Paclitaxel

NCT ID: NCT01192165

Last Updated: 2017-11-13

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

169 participants

Study Classification

INTERVENTIONAL

Study Start Date

2010-09-14

Study Completion Date

2013-10-07

Brief Summary

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The purpose of this study is to determine what dose of GSK1120212 can be given safely in combination with at least one other drug that is already approved to treat cancer. This study will test the safety of up to 6 different GSK1120212 study treatment combinations (GSK1120212 plus either docetaxel, erlotinib, pemetrexed, pemetrexed + carboplatin, pemetrexed + cisplatin, or nab-paclitaxel). The doses identified in this study may be used in future trials to test whether the combination treatment is a safe and effective therapy for subjects with metastatic lung and/or pancreatic cancers.

Detailed Description

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Conditions

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Cancer

Keywords

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Taxotere Cisplatin Carboplatin Trametinib GSK1120212 Tarceva KRAS Pemetrexed MEK inhibitor nab-Paclitaxel Docetaxel Alimta Abraxane Erlotinib

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Treatment Group 1

Trametinib plus Docetaxel

Group Type EXPERIMENTAL

Trametinib (GSK1120212)

Intervention Type DRUG

Investigational small molecule targeted therapy (MEK1/2 inhibitor)

Docetaxel

Intervention Type DRUG

Chemotherapy

Treatment Group 2

Trametinib plus Erlotinib

Group Type EXPERIMENTAL

Trametinib (GSK1120212)

Intervention Type DRUG

Investigational small molecule targeted therapy (MEK1/2 inhibitor)

Erlotinib

Intervention Type DRUG

Small molecule targeted therapy (EGFR inhibitor)

Treatment Group 3

Trametinib plus Pemetrexed

Group Type EXPERIMENTAL

Trametinib (GSK1120212)

Intervention Type DRUG

Investigational small molecule targeted therapy (MEK1/2 inhibitor)

Pemetrexed

Intervention Type DRUG

Chemotherapy

Treatment Group 4

Trametinib plus Pemetrexed and Carboplatin

Group Type EXPERIMENTAL

Trametinib (GSK1120212)

Intervention Type DRUG

Investigational small molecule targeted therapy (MEK1/2 inhibitor)

Pemetrexed

Intervention Type DRUG

Chemotherapy

Carboplatin

Intervention Type DRUG

Chemotherapy

Treatment Group 5

Trametinib plus nab-Paclitaxel

Group Type EXPERIMENTAL

Trametinib (GSK1120212)

Intervention Type DRUG

Investigational small molecule targeted therapy (MEK1/2 inhibitor)

nab-Paclitaxel

Intervention Type DRUG

Chemotherapy

Treatment Group 6

Trametinib plus Pemetrexed and Cisplatin

Group Type EXPERIMENTAL

Trametinib (GSK1120212)

Intervention Type DRUG

Investigational small molecule targeted therapy (MEK1/2 inhibitor)

Pemetrexed

Intervention Type DRUG

Chemotherapy

Cisplatin

Intervention Type DRUG

Chemotherapy

Interventions

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Trametinib (GSK1120212)

Investigational small molecule targeted therapy (MEK1/2 inhibitor)

Intervention Type DRUG

Docetaxel

Chemotherapy

Intervention Type DRUG

Erlotinib

Small molecule targeted therapy (EGFR inhibitor)

Intervention Type DRUG

Pemetrexed

Chemotherapy

Intervention Type DRUG

Carboplatin

Chemotherapy

Intervention Type DRUG

nab-Paclitaxel

Chemotherapy

Intervention Type DRUG

Cisplatin

Chemotherapy

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* The subject has a solid tumor. Expansion cohorts are limited to non-small cell lung cancer and/or pancreatic cancer with or without a KRAS mutation.
* Tumor progression following at least one prior standard therapy, the subject refuses standard therapy, or no standard therapy exists.
* The subject has a radiographically measurable tumor.
* The subject is able to carry out daily life activities without difficulty.
* The subject is able to swallow and retain oral medication.
* The subject does not have significant side effects from previous anti-cancer treatment.
* The subject has adequate organ and blood cell counts.
* Sexually active subjects must use medically acceptable methods of contraception during the course of the study.

Exclusion Criteria

* The subject has had major surgery or received certain types of cancer therapy within 2-3 weeks before starting the study.
* The subject has a brain tumor.
* Current severe, uncontrolled systemic disease.
* History of clinically significant heart, lung, or eye/vision problems.
* The subject has high blood pressure that is not well-controlled with medication.
* The subject has a permanent pacemaker.
* The subject is pregnant or breastfeeding.
* Positive for Hepatitis B, Hepatitis C, or HIV.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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GlaxoSmithKline

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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GSK Clinical Trials

Role: STUDY_DIRECTOR

GlaxoSmithKline

Locations

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GSK Investigational Site

Scottsdale, Arizona, United States

Site Status

GSK Investigational Site

Duarte, California, United States

Site Status

GSK Investigational Site

Sacramento, California, United States

Site Status

GSK Investigational Site

Denver, Colorado, United States

Site Status

GSK Investigational Site

Las Vegas, Nevada, United States

Site Status

GSK Investigational Site

Albany, New York, United States

Site Status

GSK Investigational Site

Greenville, South Carolina, United States

Site Status

GSK Investigational Site

Nashville, Tennessee, United States

Site Status

GSK Investigational Site

Dallas, Texas, United States

Site Status

GSK Investigational Site

Houston, Texas, United States

Site Status

GSK Investigational Site

Tyler, Texas, United States

Site Status

GSK Investigational Site

Norfolk, Virginia, United States

Site Status

GSK Investigational Site

Vancouver, Washington, United States

Site Status

GSK Investigational Site

Toronto, Ontario, Canada

Site Status

GSK Investigational Site

Caen, , France

Site Status

GSK Investigational Site

Marseille, , France

Site Status

GSK Investigational Site

Saint-Herblain, , France

Site Status

GSK Investigational Site

Toulouse, , France

Site Status

GSK Investigational Site

Seoul, , South Korea

Site Status

GSK Investigational Site

Seoul, , South Korea

Site Status

Countries

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United States Canada France South Korea

References

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Gandara DR, Leighl N, Delord JP, Barlesi F, Bennouna J, Zalcman G, Infante JR, Reckamp KL, Kelly K, Shepherd FA, Mazieres J, Janku F, Gardner OS, Mookerjee B, Wu Y, Cox DS, Schramek D, Peddareddigari V, Liu Y, D'Amelio AM Jr, Blumenschein G Jr. A Phase 1/1b Study Evaluating Trametinib Plus Docetaxel or Pemetrexed in Patients With Advanced Non-Small Cell Lung Cancer. J Thorac Oncol. 2017 Mar;12(3):556-566. doi: 10.1016/j.jtho.2016.11.2218. Epub 2016 Nov 19.

Reference Type DERIVED
PMID: 27876675 (View on PubMed)

Other Identifiers

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2012-000257-32

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

113486

Identifier Type: -

Identifier Source: org_study_id