Trial Outcomes & Findings for Hepatic Safety of Raltegravir Versus Efavirenz as HIV Therapy for Patients With HIV and HCV Coinfection (NCT NCT01147107)

NCT ID: NCT01147107

Last Updated: 2021-08-13

Results Overview

To estimate the rates of grade 2\*and higher ALT elevations in the two regimens.

Recruitment status

COMPLETED

Study phase

PHASE4

Target enrollment

80 participants

Primary outcome timeframe

over week 72

Results posted on

2021-08-13

Participant Flow

Participant milestones

Participant milestones
Measure
Raltegravir Based Therapy
Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Raltegravir 400 mg twice daily Raltegravir: Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Raltegravir 400 mg twice daily
Efavirenz Based Therapy
Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Efavirenz 600 mg po daily Efavirenz: Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Efavirenz 600 mg po daily
Overall Study
STARTED
39
41
Overall Study
COMPLETED
33
40
Overall Study
NOT COMPLETED
6
1

Reasons for withdrawal

Reasons for withdrawal
Measure
Raltegravir Based Therapy
Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Raltegravir 400 mg twice daily Raltegravir: Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Raltegravir 400 mg twice daily
Efavirenz Based Therapy
Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Efavirenz 600 mg po daily Efavirenz: Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Efavirenz 600 mg po daily
Overall Study
Lack of Efficacy
5
0
Overall Study
Withdrawal by Subject
1
1

Baseline Characteristics

Hepatic Safety of Raltegravir Versus Efavirenz as HIV Therapy for Patients With HIV and HCV Coinfection

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Raltegravir Based Therapy
n=38 Participants
Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Raltegravir 400 mg twice daily Raltegravir: Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Raltegravir 400 mg twice daily
Efavirenz Based Therapy
n=41 Participants
Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Efavirenz 600 mg po daily Efavirenz: Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Efavirenz 600 mg po daily
Total
n=79 Participants
Total of all reporting groups
Age, Continuous
32 years
n=5 Participants
33 years
n=7 Participants
32 years
n=5 Participants
Sex: Female, Male
Female
6 Participants
n=5 Participants
4 Participants
n=7 Participants
10 Participants
n=5 Participants
Sex: Female, Male
Male
32 Participants
n=5 Participants
37 Participants
n=7 Participants
69 Participants
n=5 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Asian
38 Participants
n=5 Participants
41 Participants
n=7 Participants
79 Participants
n=5 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Black or African American
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
White
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Region of Enrollment
Vietnam
38 participants
n=5 Participants
41 participants
n=7 Participants
79 participants
n=5 Participants

PRIMARY outcome

Timeframe: over week 72

To estimate the rates of grade 2\*and higher ALT elevations in the two regimens.

Outcome measures

Outcome measures
Measure
Raltegravir Based Therapy
n=38 Participants
Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Raltegravir 400 mg twice daily Raltegravir: Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Raltegravir 400 mg twice daily
Efavirenz Based Therapy
n=41 Participants
Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Efavirenz 600 mg po daily Efavirenz: Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Efavirenz 600 mg po daily
Rates of Grade 2 and Higher Alanine Aminotransferase (ALT) Elevations
24 Participants
30 Participants

Adverse Events

Raltegravir Based Therapy

Serious events: 8 serious events
Other events: 21 other events
Deaths: 2 deaths

Efavirenz Based Therapy

Serious events: 8 serious events
Other events: 29 other events
Deaths: 3 deaths

Serious adverse events

Serious adverse events
Measure
Raltegravir Based Therapy
n=38 participants at risk
Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Raltegravir 400 mg twice daily Raltegravir: Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Raltegravir 400 mg twice daily
Efavirenz Based Therapy
n=41 participants at risk
Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Efavirenz 600 mg po daily Efavirenz: Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Efavirenz 600 mg po daily
Injury, poisoning and procedural complications
Car Accident
2.6%
1/38 • Number of events 1 • 72 weeks
0.00%
0/41 • 72 weeks
General disorders
Suicide
0.00%
0/38 • 72 weeks
2.4%
1/41 • Number of events 1 • 72 weeks
Respiratory, thoracic and mediastinal disorders
Tuberculosis
2.6%
1/38 • Number of events 1 • 72 weeks
7.3%
3/41 • Number of events 3 • 72 weeks
Gastrointestinal disorders
Infectious Diarrhea
0.00%
0/38 • 72 weeks
2.4%
1/41 • Number of events 1 • 72 weeks
Nervous system disorders
CNS Syndrome Unclear Etiology
0.00%
0/38 • 72 weeks
2.4%
1/41 • Number of events 1 • 72 weeks
Respiratory, thoracic and mediastinal disorders
PCP Pneumonia
2.6%
1/38 • Number of events 1 • 72 weeks
0.00%
0/41 • 72 weeks
Blood and lymphatic system disorders
Lymphadenitis
2.6%
1/38 • Number of events 1 • 72 weeks
0.00%
0/41 • 72 weeks
Gastrointestinal disorders
Appendicitis
0.00%
0/38 • 72 weeks
2.4%
1/41 • Number of events 1 • 72 weeks
Renal and urinary disorders
Pyelonephritis
2.6%
1/38 • Number of events 1 • 72 weeks
0.00%
0/41 • 72 weeks
Respiratory, thoracic and mediastinal disorders
Bacterial Pneumonia
2.6%
1/38 • Number of events 1 • 72 weeks
0.00%
0/41 • 72 weeks
Nervous system disorders
PML
0.00%
0/38 • 72 weeks
2.4%
1/41 • Number of events 1 • 72 weeks
Hepatobiliary disorders
Hepatic Encephalopathy
2.6%
1/38 • Number of events 1 • 72 weeks
0.00%
0/41 • 72 weeks
Infections and infestations
Septic Shock
2.6%
1/38 • Number of events 1 • 72 weeks
0.00%
0/41 • 72 weeks

Other adverse events

Other adverse events
Measure
Raltegravir Based Therapy
n=38 participants at risk
Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Raltegravir 400 mg twice daily Raltegravir: Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Raltegravir 400 mg twice daily
Efavirenz Based Therapy
n=41 participants at risk
Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Efavirenz 600 mg po daily Efavirenz: Emtricitabine/tenofovir DF\* 200 mg/300 mg po daily + Efavirenz 600 mg po daily
Hepatobiliary disorders
ALT Elevation
55.3%
21/38 • 72 weeks
70.7%
29/41 • 72 weeks

Additional Information

Dr. Cecilia Shikuma

University of Hawaii at Manoa John A Burns School of Medicine

Phone: 8086921328

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place