Trial Outcomes & Findings for Bioequivalency Study of Imipramine Pamoate 75 mg Capsules Under Fasted Conditions (NCT NCT01107353)

NCT ID: NCT01107353

Last Updated: 2018-02-05

Results Overview

Blood samples were collected pre-dose and at intervals over 120 hours after each dose

Recruitment status

COMPLETED

Study phase

NA

Target enrollment

39 participants

Primary outcome timeframe

33 Days

Results posted on

2018-02-05

Participant Flow

Participant milestones

Participant milestones
Measure
First Imipramine Pamoate, Then Tofranil-PM
First 75 mg imipramine pamoate capsule, then 75 mg Tofranil-PM capsule (after washout period) Imipramine Pamoate: 75 mg capsule
First Tofranil PM, Then Imipramine Pamoate
First 75 mg Tofranil-PM capsule, then 75 mg imipramine pamoate capsule (after washout period) Imipramine Pamoate: 75 mg capsule
Overall Study
STARTED
20
20
Overall Study
COMPLETED
19
20
Overall Study
NOT COMPLETED
1
0

Reasons for withdrawal

Reasons for withdrawal
Measure
First Imipramine Pamoate, Then Tofranil-PM
First 75 mg imipramine pamoate capsule, then 75 mg Tofranil-PM capsule (after washout period) Imipramine Pamoate: 75 mg capsule
First Tofranil PM, Then Imipramine Pamoate
First 75 mg Tofranil-PM capsule, then 75 mg imipramine pamoate capsule (after washout period) Imipramine Pamoate: 75 mg capsule
Overall Study
Positive Drug Screen
1
0

Baseline Characteristics

Bioequivalency Study of Imipramine Pamoate 75 mg Capsules Under Fasted Conditions

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
First Imipramine Pamoate, Then Tofranil-PM
n=20 Participants
First 75 mg imipramine pamoate capsule, then 75 mg Tofranil-PM capsule (after washout period) Imipramine Pamoate: 75 mg capsule
First Tofranil PM, Then Imipramine Pamoate
n=20 Participants
First 75 mg Tofranil-PM capsule, then 75 mg imipramine pamoate capsule (after washout period) Imipramine Pamoate: 75 mg capsule
Total
n=40 Participants
Total of all reporting groups
Age, Continuous
28.41 years
STANDARD_DEVIATION 7.65 • n=5 Participants
28.41 years
STANDARD_DEVIATION 7.65 • n=7 Participants
28.41 years
STANDARD_DEVIATION 7.65 • n=5 Participants
Sex: Female, Male
Female
6 Participants
n=5 Participants
7 Participants
n=7 Participants
13 Participants
n=5 Participants
Sex: Female, Male
Male
14 Participants
n=5 Participants
13 Participants
n=7 Participants
27 Participants
n=5 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Asian
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Black or African American
19 Participants
n=5 Participants
17 Participants
n=7 Participants
36 Participants
n=5 Participants
Race (NIH/OMB)
White
0 Participants
n=5 Participants
3 Participants
n=7 Participants
3 Participants
n=5 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Race (NIH/OMB)
Unknown or Not Reported
1 Participants
n=5 Participants
0 Participants
n=7 Participants
1 Participants
n=5 Participants
Region of Enrollment
United States
20 participants
n=5 Participants
20 participants
n=7 Participants
40 participants
n=5 Participants

PRIMARY outcome

Timeframe: 33 Days

Blood samples were collected pre-dose and at intervals over 120 hours after each dose

Outcome measures

Outcome measures
Measure
First Imipramine Pamoate, Then Tofranil-PM
n=19 Participants
First 75 mg imipramine pamoate capsule, then 75 mg Tofranil-PM capsule (after washout period) Imipramine Pamoate: 75 mg capsule
First Tofranil PM, Then Imipramine Pamoate
n=19 Participants
First 75 mg Tofranil-PM capsule, then 75 mg imipramine pamoate capsule (after washout period) Imipramine Pamoate: 75 mg capsule
Bioequivalence Determined by Statistical Comparison Cmax
11.5 ng/mL
Standard Deviation 7.48
11.3 ng/mL
Standard Deviation 7.03

Adverse Events

First Imipramine Pamoate, Then Tofranil-PM

Serious events: 0 serious events
Other events: 0 other events
Deaths: 0 deaths

First Tofranil PM, Then Imipramine Pamoate

Serious events: 0 serious events
Other events: 0 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Adverse event data not reported

Additional Information

Anton (Tony) Amann, PhD., Executive Director, DRAMA

Roxane Laboratories, Inc.

Phone: 614-272-4785

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place

Restriction type: GT60