BAY80-6946 Open Label, Phase I Study in Patients With Advanced Cancer

NCT ID: NCT00962611

Last Updated: 2017-10-06

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

57 participants

Study Classification

INTERVENTIONAL

Study Start Date

2009-11-19

Study Completion Date

2016-02-23

Brief Summary

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The purpose of this study is to determine the tolerability, maximum tolerated dose and pharmacokinetics of this drug.

Detailed Description

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Conditions

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Neoplasms

Study Design

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Allocation Method

NA

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Copanlisib

Group Type EXPERIMENTAL

Copanlisib (Aliqopa, BAY80-6946)

Intervention Type DRUG

BAY80-6946 given IV over 1 hour every week for three weeks with a one week break until progression or unacceptable toxicities develop.

Interventions

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Copanlisib (Aliqopa, BAY80-6946)

BAY80-6946 given IV over 1 hour every week for three weeks with a one week break until progression or unacceptable toxicities develop.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Age \>/= 18 years.
* Histological or cytological documentation of non-hematologic, malignant solid tumor, excluding primary brain or spinal tumors, or history of central nervous system metastases
* At least one measurable lesion or evaluable disease
* Life expectancy of at least 12 weeks
* ECOG Performance Status of 0, 1 or 2
* PT-INR/PTT \< 1.5 x upper limit of normal \[Patients who are being therapeutically anticoagulated with an agent such as coumadin or heparin will be allowed to participate provided that no prior evidence of underlying abnormality in these parameters exists\]. Low-dose aspirin is permitted (\</= 100 mg daily).
* Adequate bone marrow, liver and renal function
* Ability to understand and to sign an informed consent form; a signed informed consent must be obtained prior to any study specific procedures

Exclusion Criteria

* History of cardiac disease congestive heart failure (CHF) \> NYHA Class II; active coronary artery disease, myocardial infarction within 6 months prior to study entry; new onset angina within 3 months prior to study entry or unstable angina or cardiac arrhythmias requiring anti-arrhythmic therapy (beta-blockers or Digoxin are permitted).
* Current diagnosis of type I or II diabetes mellitus or fasting blood glucose level \>125 mg/dL at screening, or HbA1c 7%
* Active clinically serious infections \> Grade 2 (NCI-CTCAE Version 3.0)
* History of having received allogeneic organ transplant
* Uncontrolled seizure disorder. Use of cytochrome P450 enzyme-inducing antiepileptic drugs (phenytoin, carbamazepine or phenobarbital) is not allowed throughout the entire study.
* Uncontrolled hypertension defined as systolic blood pressure \> 150 mmHg or diastolic pressure \> 90 mmHg, despite optimal medical management
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Bayer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Bayer Study Director

Role: STUDY_DIRECTOR

Bayer

Locations

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Scottsdale, Arizona, United States

Site Status

Pittsburgh, Pennsylvania, United States

Site Status

San Antonio, Texas, United States

Site Status

Countries

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United States

References

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A. Patnaik et al. Supplementary materials /Supplementary methods. Annals of Oncology 2016

Reference Type BACKGROUND

Rowe EL. Automated drop volume apparatus for surface tension measurement. J Pharm Sci. 1972 May;61(5):781-2. doi: 10.1002/jps.2600610523. No abstract available.

Reference Type RESULT
PMID: 5035790 (View on PubMed)

Patnaik A, Appleman LJ, Tolcher AW, Papadopoulos KP, Beeram M, Rasco DW, Weiss GJ, Sachdev JC, Chadha M, Fulk M, Ejadi S, Mountz JM, Lotze MT, Toledo FG, Chu E, Jeffers M, Pena C, Xia C, Reif S, Genvresse I, Ramanathan RK. First-in-human phase I study of copanlisib (BAY 80-6946), an intravenous pan-class I phosphatidylinositol 3-kinase inhibitor, in patients with advanced solid tumors and non-Hodgkin's lymphomas. Ann Oncol. 2016 Oct;27(10):1928-40. doi: 10.1093/annonc/mdw282.

Reference Type DERIVED
PMID: 27672108 (View on PubMed)

Other Identifiers

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12871

Identifier Type: -

Identifier Source: org_study_id