Trial Outcomes & Findings for Ropinirole 0.25 mg Tablets Under Fasting Conditions (NCT NCT00829504)

NCT ID: NCT00829504

Last Updated: 2009-09-11

Results Overview

Bioequivalence based on Cmax.

Recruitment status

COMPLETED

Study phase

PHASE1

Target enrollment

44 participants

Primary outcome timeframe

Blood samples collected over a 24 hour period.

Results posted on

2009-09-11

Participant Flow

Participant milestones

Participant milestones
Measure
Test (Ropinirole HCl) First
0.25 mg Ropinirole HCl Tablets test product dosed in first period followed by 0.25 mg Requip® Tablets reference product dosed in the second period.
Reference (Requip®) First
0.25 mg Requip® Tablets reference product dosed in first period followed by 0.25 mg Ropinirole HCl Tablets test product dosed in the second period.
First Intervention
STARTED
22
22
First Intervention
COMPLETED
21
22
First Intervention
NOT COMPLETED
1
0
Washout of 7 Days
STARTED
21
22
Washout of 7 Days
COMPLETED
20
22
Washout of 7 Days
NOT COMPLETED
1
0
Second Intervention
STARTED
20
22
Second Intervention
COMPLETED
19
22
Second Intervention
NOT COMPLETED
1
0

Reasons for withdrawal

Reasons for withdrawal
Measure
Test (Ropinirole HCl) First
0.25 mg Ropinirole HCl Tablets test product dosed in first period followed by 0.25 mg Requip® Tablets reference product dosed in the second period.
Reference (Requip®) First
0.25 mg Requip® Tablets reference product dosed in first period followed by 0.25 mg Ropinirole HCl Tablets test product dosed in the second period.
First Intervention
Adverse Event
1
0
Washout of 7 Days
Withdrawal by Subject
1
0
Second Intervention
Physician Decision
1
0

Baseline Characteristics

Ropinirole 0.25 mg Tablets Under Fasting Conditions

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Test (Ropinirole HCl) First
n=22 Participants
0.25 mg Ropinirole HCl Tablets test product dosed in first period followed by 0.25 mg Requip® Tablets reference product dosed in the second period.
Reference (Requip®) First
n=22 Participants
0.25 mg Requip® Tablets reference product dosed in first period followed by 0.25 mg Ropinirole HCl Tablets test product dosed in the second period.
Total
n=44 Participants
Total of all reporting groups
Age, Categorical
<=18 years
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Age, Categorical
Between 18 and 65 years
22 Participants
n=5 Participants
22 Participants
n=7 Participants
44 Participants
n=5 Participants
Age, Categorical
>=65 years
0 Participants
n=5 Participants
0 Participants
n=7 Participants
0 Participants
n=5 Participants
Sex: Female, Male
Female
5 Participants
n=5 Participants
10 Participants
n=7 Participants
15 Participants
n=5 Participants
Sex: Female, Male
Male
17 Participants
n=5 Participants
12 Participants
n=7 Participants
29 Participants
n=5 Participants
Race/Ethnicity, Customized
Black
13 participants
n=5 Participants
17 participants
n=7 Participants
30 participants
n=5 Participants
Race/Ethnicity, Customized
White
0 participants
n=5 Participants
1 participants
n=7 Participants
1 participants
n=5 Participants
Race/Ethnicity, Customized
Hispanic
9 participants
n=5 Participants
4 participants
n=7 Participants
13 participants
n=5 Participants
Region of Enrollment
United States
22 participants
n=5 Participants
22 participants
n=7 Participants
44 participants
n=5 Participants

PRIMARY outcome

Timeframe: Blood samples collected over a 24 hour period.

Population: All participants that completed the study had their samples analyzed.

Bioequivalence based on Cmax.

Outcome measures

Outcome measures
Measure
Test (Ropinirole HCl)
n=40 Participants
0.25 mg Ropinirole HCl Tablets test product dosed in either period.
Reference (Requip®)
n=40 Participants
0.25 mg Requip® Tablets reference product dosed in either period.
Cmax (Maximum Observed Concentration of Drug Substance in Plasma)
552.1 pg/mL
Standard Deviation 219.01
546.5 pg/mL
Standard Deviation 205.72

PRIMARY outcome

Timeframe: Blood samples collected over a 24 hour period.

Population: All participants that completed the study had their samples analyzed.

Bioequivalence based on AUC0-t.

Outcome measures

Outcome measures
Measure
Test (Ropinirole HCl)
n=40 Participants
0.25 mg Ropinirole HCl Tablets test product dosed in either period.
Reference (Requip®)
n=40 Participants
0.25 mg Requip® Tablets reference product dosed in either period.
AUC0-t (Area Under the Concentration-time Curve From Time Zero to Time of Last Measurable Concentration)
4190.92 pg*h/mL
Standard Deviation 2290.13
4062.99 pg*h/mL
Standard Deviation 2073.39

PRIMARY outcome

Timeframe: Blood samples collected over a 24 hour period.

Population: All participants that completed the study had their samples analyzed.

Bioequivalence based on AUC0-inf.

Outcome measures

Outcome measures
Measure
Test (Ropinirole HCl)
n=40 Participants
0.25 mg Ropinirole HCl Tablets test product dosed in either period.
Reference (Requip®)
n=40 Participants
0.25 mg Requip® Tablets reference product dosed in either period.
AUC0-inf (Area Under the Concentration-time Curve From Time Zero to Infinity)
4469 pg*h/mL
Standard Deviation 2561.37
4305.88 pg*h/mL
Standard Deviation 2283.55

Adverse Events

Serious adverse events

Adverse event data not reported

Other adverse events

Adverse event data not reported

Additional Information

Manager, Biopharmaceutics

TEVA Pharmaceuticals, USA

Phone: 1-866-384-5525

Results disclosure agreements

  • Principal investigator is a sponsor employee The Principal Investigator is not permitted to discuss or publish trial results.
  • Publication restrictions are in place

Restriction type: OTHER