Pharmacokinetics, Safety And Toleration Of Maraviroc Administered To Subjects With Various Degrees Of Renal Impaired And Normal Renal Function

NCT ID: NCT00717067

Last Updated: 2010-11-19

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE4

Total Enrollment

30 participants

Study Classification

INTERVENTIONAL

Study Start Date

2008-07-31

Study Completion Date

2008-11-30

Brief Summary

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The purpose of this study is to assess whether a dosing adjustment is needed in patients with renal impairment.

Detailed Description

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Conditions

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Human Immunodeficiency Virus (HIV) Infection

Keywords

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maraviroc, pharmacokinetics, renal impairment

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Healthy Subjects

Subjects with Normal Renal Function (Creatinine Clearance \> 80mL/min) (I) Maraviroc single dose, followed by (II) Maraviroc + Saquinavir/Ritonavir

Group Type EXPERIMENTAL

Maraviroc

Intervention Type DRUG

Maraviroc 300 mg (150 mg x 2 tablets) x single dose

Maraviroc

Intervention Type DRUG

Maraviroc 150 mg tablet twice daily x 7 days

Ritonavir

Intervention Type DRUG

Ritonavir 100 mg capsule twice daily x 7 days

Saquinavir

Intervention Type DRUG

Saquinavir 1000 mg (500 mg x 2 tablets) twice daily x 7 days

Mild Renal Impairment

Subjects with Mild Renal Impairment (Creatinine Clearance \>50 and ≤80 mL/min)

Group Type EXPERIMENTAL

Maraviroc

Intervention Type DRUG

Maraviroc 150 mg tablet once daily x 7 days

Ritonavir

Intervention Type DRUG

Ritonavir 100 mg capsule twice daily x 7 days

Saquinavir

Intervention Type DRUG

Saquinavir 1000 mg (500 mg x 2 tablets) twice daily x 7 days

Moderate Renal Impairment

Subjects with Moderate Renal Impairment (Creatinine Clearance ≥30 and ≤50 mL/min)

Group Type EXPERIMENTAL

Maraviroc

Intervention Type DRUG

Maraviroc 150 mg tablet once every 48 hours x 7 days

Ritonavir

Intervention Type DRUG

Ritonavir 100 mg capsule twice daily x 7 days

Saquinavir

Intervention Type DRUG

Saquinavir 1000 mg (500 mg x 2 tablets) twice daily x 7 days

Severe Renal Impairment

Subjects with Severe Renal Impairment (Creatinine Clearance \<30 mL/min)

Group Type EXPERIMENTAL

Maraviroc

Intervention Type DRUG

Maraviroc 300 mg (150 mg x 2 tablets) x single dose

ESRD on Hemodialysis

Subjects with End Stage Renal Impairment receiving Hemodialysis(Creatinine Clearance \<30 mL/min) (I) Maraviroc single dose one hour following completion of hemodialysis, followed by (II) Maraviroc single dose three hours prior to start of hemodialysis

Group Type EXPERIMENTAL

Maraviroc

Intervention Type DRUG

Maraviroc 300 mg (150 mg x 2 tablets) x single dose one hour following completion of hemodialysis

Maraviroc

Intervention Type DRUG

Maraviroc 300 mg (150 mg x 2 tablets) x single dose three hours prior to start of hemodialysis

Interventions

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Maraviroc

Maraviroc 300 mg (150 mg x 2 tablets) x single dose

Intervention Type DRUG

Maraviroc

Maraviroc 150 mg tablet twice daily x 7 days

Intervention Type DRUG

Ritonavir

Ritonavir 100 mg capsule twice daily x 7 days

Intervention Type DRUG

Saquinavir

Saquinavir 1000 mg (500 mg x 2 tablets) twice daily x 7 days

Intervention Type DRUG

Maraviroc

Maraviroc 150 mg tablet once daily x 7 days

Intervention Type DRUG

Ritonavir

Ritonavir 100 mg capsule twice daily x 7 days

Intervention Type DRUG

Saquinavir

Saquinavir 1000 mg (500 mg x 2 tablets) twice daily x 7 days

Intervention Type DRUG

Maraviroc

Maraviroc 150 mg tablet once every 48 hours x 7 days

Intervention Type DRUG

Ritonavir

Ritonavir 100 mg capsule twice daily x 7 days

Intervention Type DRUG

Saquinavir

Saquinavir 1000 mg (500 mg x 2 tablets) twice daily x 7 days

Intervention Type DRUG

Maraviroc

Maraviroc 300 mg (150 mg x 2 tablets) x single dose

Intervention Type DRUG

Maraviroc

Maraviroc 300 mg (150 mg x 2 tablets) x single dose one hour following completion of hemodialysis

Intervention Type DRUG

Maraviroc

Maraviroc 300 mg (150 mg x 2 tablets) x single dose three hours prior to start of hemodialysis

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Stable Renal Function defined as ≤20% (25% for normal renal function) difference between 2 measurements of serum creatinine obtained on 2 occasions separated by at least 2 weeks.
* Body Mass Index (BMI) of approximately 18 to 40 kg/m2 inclusive.
* Total body weight \>50 kg (110 lbs).
* Male or female subjects between the ages of 18 and 85 years.

Exclusion Criteria

* Subjects with acute renal disease and/or history of renal transplant.
* Supine BP at Screening ≥160 mm Hg systolic or ≥95 mm Hg diastolic.
* Supine BP at Screening ≤80 mm Hg systolic or ≤40 mm Hg diastolic.
Minimum Eligible Age

18 Years

Maximum Eligible Age

85 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Pfizer

INDUSTRY

Sponsor Role collaborator

ViiV Healthcare

INDUSTRY

Sponsor Role lead

Responsible Party

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Pfizer, Inc.

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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Pfizer Investigational Site

Berlin, , Germany

Site Status

Pfizer Investigational Site

München, , Germany

Site Status

Countries

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Germany

Related Links

Other Identifiers

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A4001075

Identifier Type: -

Identifier Source: org_study_id