A Study of SB-742457, Added to Donepezil for the Treatment of Mild-to-moderate Alzheimer's Disease

NCT ID: NCT00710684

Last Updated: 2017-12-07

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

682 participants

Study Classification

INTERVENTIONAL

Study Start Date

2008-07-01

Study Completion Date

2010-11-16

Brief Summary

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The study is designed to investigate the safety and efficacy of SB-742457 when added to stable donepezil treatment in subjects with mild-to-moderate Alzheimer's disease.

Detailed Description

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Conditions

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Alzheimer's Disease

Keywords

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Alzheimer's disease cognition SB-742457

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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DONEPEZIL + SB-742457 15 MG

SB-742457 - 15mg added to existing donepezil treatment

Group Type EXPERIMENTAL

SB-742457 15mg

Intervention Type DRUG

SB-742457 - 15mg added to existing donepezil treatment

donepezil 5-10mg

Intervention Type DRUG

existing donepezil treatment

DONEPEZIL + PLACEBO

Placebo added to existing donepezil

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Placebo added to existing donepezil

donepezil 5-10mg

Intervention Type DRUG

existing donepezil treatment

DONEPEZIL + SB-742457 35 MG

SB-742457 - 35mg added to existing donepezil

Group Type EXPERIMENTAL

SB-742457 35mg

Intervention Type DRUG

SB-742457 - 35mg added to existing donepezil

donepezil 5-10mg

Intervention Type DRUG

existing donepezil treatment

Interventions

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SB-742457 15mg

SB-742457 - 15mg added to existing donepezil treatment

Intervention Type DRUG

SB-742457 35mg

SB-742457 - 35mg added to existing donepezil

Intervention Type DRUG

Placebo

Placebo added to existing donepezil

Intervention Type DRUG

donepezil 5-10mg

existing donepezil treatment

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Subjects and their caregivers must provide informed consent prior to study entry.
* Subjects must have a clinical diagnosis of probable mild-to-moderate Alzheimer's disease with no evidence of disorders that are thought to be the cause of, or contributing to the severity of the subject's dementia and a documented history of at least 6 months of ongoing donepezil therapy with stable dosing for at least the last 2 months.
* Subjects must have a regular caregiver who is willing to attend visits, oversee the subject's compliance with the study and report on the subject's status.
* Female subjects of child-bearing potential must agree to abstinence or an approved form of birth control.
* Subjects must have adequate blood pressure and laboratory values.

Exclusion Criteria

* Subjects with a diagnosis of possible, probable or definite vascular dementia may not participate.
* Subjects with known hypersensitivity to sunlight or a history of seizures, previous exposure to SB-742457, taking agents for which there is a theoretical risk of interaction with SB-742457, or taking medication for Alzheimer's disease or centrally acting agents which might impact study outcomes may not participate.
Minimum Eligible Age

50 Years

Maximum Eligible Age

85 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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GlaxoSmithKline

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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GSK Clinical Trials

Role: STUDY_DIRECTOR

GlaxoSmithKline

Locations

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GSK Investigational Site

Litchfield Park, Arizona, United States

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Fresno, California, United States

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Rancho Mirage, California, United States

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San Francisco, California, United States

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Hallandale, Florida, United States

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Hialeah, Florida, United States

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Paterson, New Jersey, United States

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Syracuse, New York, United States

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Winston-Salem, North Carolina, United States

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Columbus, Ohio, United States

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Tulsa, Oklahoma, United States

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Memphis, Tennessee, United States

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Austin, Texas, United States

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Bennington, Vermont, United States

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Ciudad Autonoma de Buenos Aires, Buenos Aires, Argentina

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Ciudad Autonoma de Buenos Aires, Buenos Aires, Argentina

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Ciudad de Buenos Aires, Buenos Aires, Argentina

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La Plata, Buenos Aires, Argentina

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Córdoba, Córdoba Province, Argentina

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Buenos Aires, , Argentina

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Santa Fe, , Argentina

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Kogarah, New South Wales, Australia

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Herston, Queensland, Australia

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Woodville, South Australia, Australia

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Ballarat, Victoria, Australia

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Heidelberg West, Victoria, Australia

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Kew, Victoria, Australia

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Nedlands, Western Australia, Australia

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Saint John, New Brunswick, Canada

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Kentville, Nova Scotia, Canada

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Ottawa, Ontario, Canada

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Peterborough, Ontario, Canada

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Toronto, Ontario, Canada

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Toronto, Ontario, Canada

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Greenfield Park, Quebec, Canada

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Montreal, Quebec, Canada

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Sherbrooke, Quebec, Canada

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Sherbrooke, Quebec, Canada

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Québec, , Canada

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Viña del Mar, Región de Valparaíso, Chile

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Santiago, Región Metro de Santiago, Chile

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Santiago, Región Metro de Santiago, Chile

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Santiago, , Chile

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Mělník, , Czechia

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Olomouc, , Czechia

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Ostrava, , Czechia

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Pardubice, , Czechia

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Pilsen, , Czechia

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Prague, , Czechia

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Prague, , Czechia

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Prague, , Czechia

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Ellwangen, Baden-Wurttemberg, Germany

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Stuttgart, Baden-Wurttemberg, Germany

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Tübingen, Baden-Wurttemberg, Germany

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Ulm, Baden-Wurttemberg, Germany

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Alzenau in Unterfranken, Bavaria, Germany

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Günzburg, Bavaria, Germany

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Munich, Bavaria, Germany

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Regensburg, Bavaria, Germany

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Unterhaching, Bavaria, Germany

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Bad Homburg, Hesse, Germany

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Achim, Lower Saxony, Germany

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Schwerin, Mecklenburg-Vorpommern, Germany

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Schwerin, Mecklenburg-Vorpommern, Germany

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Aachen, North Rhine-Westphalia, Germany

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Bad Honnef, North Rhine-Westphalia, Germany

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Bochum, North Rhine-Westphalia, Germany

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Dresden, Saxony, Germany

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Dresden, Saxony, Germany

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Jena, Thuringia, Germany

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Berlin, , Germany

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Berlin, , Germany

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Berlin, , Germany

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Chieti Scalo, Abruzzo, Italy

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Napoli, Campania, Italy

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San Felice A Cancello - Caserta, Campania, Italy

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Cassino (FR), Lazio, Italy

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Rome, Lazio, Italy

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Rome, Lazio, Italy

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Brescia, Lombardy, Italy

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Castellanza (VA), Lombardy, Italy

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Milan, Lombardy, Italy

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Milan, Lombardy, Italy

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Rho, Lombardy, Italy

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Turin, Piedmont, Italy

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Lido Di Camaiore (LU), Tuscany, Italy

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Pisa, Tuscany, Italy

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Perugia, Umbria, Italy

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Valdagno (VI), Veneto, Italy

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Verona, Veneto, Italy

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Baracaldo/Vizcaya, , Spain

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Barcelona, , Spain

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Barcelona, , Spain

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Barcelona, , Spain

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Burgos, , Spain

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Castellon, , Spain

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Madrid, , Spain

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Murcia, , Spain

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Salamanca, , Spain

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San Sebastián, , Spain

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San Vicente Del Raspeig/Alicante, , Spain

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Valencia, , Spain

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Countries

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United States Argentina Australia Canada Chile Czechia Germany Italy Spain

References

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Maher-Edwards G, Watson C, Ascher J, Barnett C, Boswell D, Davies J, Fernandez M, Kurz A, Zanetti O, Safirstein B, Schronen JP, Zvartau-Hind M, Gold M. Two randomized controlled trials of SB742457 in mild-to-moderate Alzheimer's disease. Alzheimers Dement (N Y). 2015 May 7;1(1):23-36. doi: 10.1016/j.trci.2015.04.001. eCollection 2015 Jun.

Reference Type DERIVED
PMID: 29854923 (View on PubMed)

Other Identifiers

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AZ3110866

Identifier Type: -

Identifier Source: org_study_id