A Placebo Controlled Safety and Efficacy Study of INT131 Besylate in Type 2 Diabetes, With an Active Comparator

NCT ID: NCT00631007

Last Updated: 2010-09-13

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

367 participants

Study Classification

INTERVENTIONAL

Study Start Date

2008-02-29

Study Completion Date

2009-09-30

Brief Summary

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This is a 24 week study comparing the efficacy of four dose levels of INT131 besylate with pioglitazone HCl in patients with type 2 diabetes. Eligible patients will be men and women (of non-childbearing potential or using dual barrier methods of contraception) between 30 and 75 years of age who are minimally responsive to treatment with sulfonylurea monotherapy or sulfonylurea plus metformin combination therapy.

Detailed Description

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Conditions

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Type 2 Diabetes Mellitus

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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INT131 besylate 0.5 mg

INT131 besylate 0.5 mg once-daily administration and matching placebo to pioglitazone HCl.

Group Type EXPERIMENTAL

INT131 besylate

Intervention Type DRUG

Once-daily, oral

INT131 besylate 1 mg

INT131 besylate 1 mg once-daily administration and matching placebo to pioglitazone HCl

Group Type EXPERIMENTAL

INT131 besylate

Intervention Type DRUG

Once-daily, oral

INT131 besylate 2 mg

INT131 besylate 2 mg administered once-daily and matching placebo to pioglitazone HCl

Group Type EXPERIMENTAL

INT131 besylate

Intervention Type DRUG

Once-daily, oral

INT131 besylate 3 mg

INT131 besylate 3 mg administered once-daily and matching placebo to pioglitazone HCl

Group Type EXPERIMENTAL

INT131 besylate

Intervention Type DRUG

Once-daily, oral

pioglitazone HCl 45 mg

pioglitazone HCl 45 mg administered once-daily and matching placebo to INT131 besylate

Group Type ACTIVE_COMPARATOR

Pioglitazone HCl

Intervention Type DRUG

Once-daily, oral

placebo

placebo administered once-daily, matching placebo to INT131 besylate and matching placebo to pioglitazone HCl

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Once-daily, oral

Interventions

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INT131 besylate

Once-daily, oral

Intervention Type DRUG

Pioglitazone HCl

Once-daily, oral

Intervention Type DRUG

Placebo

Once-daily, oral

Intervention Type DRUG

Other Intervention Names

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Actos

Eligibility Criteria

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Inclusion Criteria

* Diagnosis of Type 2 diabetes and on either sulfonylurea monotherapy or sulfonylurea plus metformin combination therapy for at least 3 months at stable dose
* Males and Females (of non-childbearing potential or who are using dual barrier methods of contraception) between 30 and 75 years of age
* HbA1c must be ≥7.5% and ≤10% at screening
* Fasting Plasma Glucose must be \<240 mg/dL at screening

Exclusion Criteria

* History of type 1 diabetes
* History of diabetic ketoacidosis
* NYHA Class III or IV cardiac status or hospitalization for congestive heart failure within 6 weeks prior to Visit 1
* Treatment with any non-peroxisome proliferator-activated receptor (non-PPAR) antidiabetic agent, investigational or approved, other than metformin or permitted sulfonylureas within 3 months prior to screening
* Treatment with rosiglitazone, pioglitazone, or any PPAR investigational antidiabetic agent within 6 month prior to screening
* Body mass index \>45 kg/m2
* Fasting triglycerides \>500 mg/dL
* Uncontrolled hypertension (sitting systolic blood pressure \>160 mmHg and/or sitting diastolic blood pressure \>100 mmHg
* Presence of diabetic complications, which in the opinion of the investigator, would complicate the subject's participation in the study (i.e., require initiation of new medication)
Minimum Eligible Age

30 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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InteKrin Therapeutics, Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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InteKrin Therapeutics Inc.

Principal Investigators

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David Orloff, MD

Role: STUDY_DIRECTOR

Medpace, Inc.

Locations

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Northern California Research

Carmichael, California, United States

Site Status

National Research Institute

Los Angeles, California, United States

Site Status

VA San Diego Healthcare System

San Diego, California, United States

Site Status

Apex Research Institute

Santa Ana, California, United States

Site Status

Internal Medicine of the Rockies

Colorado Springs, Colorado, United States

Site Status

Creekside Endocrine Associates, PC

Denver, Colorado, United States

Site Status

Clinical Research Consulting, LLC

Milford, Connecticut, United States

Site Status

MedStar Research Institute

Washington D.C., District of Columbia, United States

Site Status

Clinical Research of South Florida

Coral Gables, Florida, United States

Site Status

The Center for Diabetes and Endocrine Care

Hollywood, Florida, United States

Site Status

Baptist Diabetes Associates, PA

Miami, Florida, United States

Site Status

International Research Associates, LLC

Miami, Florida, United States

Site Status

Elite Research Institute

Miami, Florida, United States

Site Status

Suncoast Clinical Research, Inc.

New Port Richey, Florida, United States

Site Status

Suncoast Clinical Research, Inc.

Palm Harbor, Florida, United States

Site Status

Meridien Research

Tampa, Florida, United States

Site Status

Meridien Research

Tampa, Florida, United States

Site Status

Clinical Research of Central Florida

Winter Haven, Florida, United States

Site Status

Executive Health and Research Associates, Inc.

Atlanta, Georgia, United States

Site Status

Endocrine Research Solutions, Inc.

Roswell, Georgia, United States

Site Status

Cedar-Crosse Research Center

Chicago, Illinois, United States

Site Status

ICCT Reseach International

Chicago, Illinois, United States

Site Status

American Health Network

Indianapolis, Indiana, United States

Site Status

L-Marc Research Center

Louisville, Kentucky, United States

Site Status

New Orleans Center for Clinical Research

New Orleans, Louisiana, United States

Site Status

Stephen R. Smith, MD

Baltimore, Maryland, United States

Site Status

Olive Branch Family Medical Center

Olive Branch, Mississippi, United States

Site Status

Diabetes and Endocrinology Specialists, Inc.

Chesterfield, Missouri, United States

Site Status

Saint Luke's Lipid and Diabetes Reseach Center

Kansas City, Missouri, United States

Site Status

Bozeman Deaconess Internal Medicine Associates

Bozeman, Montana, United States

Site Status

Comprehensive Clinical Research

Berlin, New Jersey, United States

Site Status

Kaleida Health Diabetes Center

Buffalo, New York, United States

Site Status

UNC Diabetes Care Center/Highgate Specialty Center

Durham, North Carolina, United States

Site Status

Fairbrook Medical Clinic

Hickory, North Carolina, United States

Site Status

Diabetes & Endrocrinology Consultants

Morehead City, North Carolina, United States

Site Status

The Lindner Clinical Trial Center

Cincinnati, Ohio, United States

Site Status

IVA Research

Cincinnati, Ohio, United States

Site Status

Rapid Medical Research, Inc

Cleveland, Ohio, United States

Site Status

Opitmed Research, LTD

Columbus, Ohio, United States

Site Status

ResEvo LLC

Cuyahoga Falls, Ohio, United States

Site Status

Delaware Smith Clinic

Delaware, Ohio, United States

Site Status

Prestige Clinical Research

Franklin, Ohio, United States

Site Status

Wells Institute for Health Awareness

Kettering, Ohio, United States

Site Status

Frederick C Smith Clinic

Marion, Ohio, United States

Site Status

Your Diabetes Endocrine Nutrition Group, LLC

Mentor, Ohio, United States

Site Status

Clinical Research Source, Inc

Perrysburg, Ohio, United States

Site Status

Tri-State Medical Group, Inc.

Beaver, Pennsylvania, United States

Site Status

Lycoming Internal Medicine, Inc.

Jersey Shore, Pennsylvania, United States

Site Status

New England Center for Clinical Research

Cranston, Rhode Island, United States

Site Status

Hartwell Research Group

Anderson, South Carolina, United States

Site Status

Medical Research South

Charleston, South Carolina, United States

Site Status

Palmetto Clinical Trial Services, LLC

Simpsonville, South Carolina, United States

Site Status

Dallas Diabetes and Endocrine Research Center

Dallas, Texas, United States

Site Status

Research Institute of Dallas

Dallas, Texas, United States

Site Status

Baylor University Endocrine Center

Dallas, Texas, United States

Site Status

Diabetes Center of the Southwest

Midland, Texas, United States

Site Status

Quality Research, Inc.

San Antonio, Texas, United States

Site Status

DGD Research

San Antonio, Texas, United States

Site Status

Salem VA Medical Center R&D Office

Salem, Virginia, United States

Site Status

Nucleo Medico Vallarta

Guadalajara, Jalisco, Mexico

Site Status

Comite Mexicano para la Prevencion de la Osteoporosis A.C.

Mexico City, Mexico DF, Mexico

Site Status

Centro Especializado en Diabetes y Obisidad (EDOPEC)

Mexico City, Mexico DF, Mexico

Site Status

Instituto Nacional de Nutricion Salvador Zubiran (INNSZ)

Mexico City, Mexico DF, Mexico

Site Status

Instituto Mexicano de Investigacion Clinica

Mexico City, Mexico DF, Mexico

Site Status

Unidad Metabolica y Cardiovascular SC

Cuernavaca, Morelos, Mexico

Site Status

Hospital Santa Engracia

Monterrey, Nuevo León, Mexico

Site Status

Countries

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United States Mexico

References

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DePaoli AM, Higgins LS, Henry RR, Mantzoros C, Dunn FL; INT131-007 Study Group. Can a selective PPARgamma modulator improve glycemic control in patients with type 2 diabetes with fewer side effects compared with pioglitazone? Diabetes Care. 2014 Jul;37(7):1918-23. doi: 10.2337/dc13-2480. Epub 2014 Apr 10.

Reference Type DERIVED
PMID: 24722496 (View on PubMed)

Other Identifiers

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INT131-007

Identifier Type: -

Identifier Source: org_study_id