Study to Evaluate Erlotinib With or Without SNDX-275 (Entinostat) in the Treatment of Patients With Advanced NSCLC

NCT ID: NCT00602030

Last Updated: 2022-08-22

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1/PHASE2

Total Enrollment

141 participants

Study Classification

INTERVENTIONAL

Study Start Date

2008-01-08

Study Completion Date

2012-02-01

Brief Summary

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The purpose of this study is to evaluate the safety and efficacy of entinostat in combination with erlotinib in the treatment of Advanced Non-Small Cell Lung Cancer (NSCLC).

Detailed Description

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Conditions

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Non-Small-Cell Lung Carcinoma Carcinoma, Non-Small Cell Lung

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

TRIPLE

Participants Caregivers Investigators

Study Groups

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Lead-in Phase: Erlotinib + Entinostat 5 mg

Erlotinib 150 mg, tablets, orally, daily plus entinostat 5 mg, tablets, orally, on Days 1 and 15 of each 28-day cycle until disease progression or intolerable toxicities for up to 6 cycles in the Lead-in Phase.

Group Type EXPERIMENTAL

Entinostat

Intervention Type DRUG

Entinostat tablets on Days 1 and 15 of a 28-day cycle.

Erlotinib

Intervention Type DRUG

Erlotinib 150 mg tablets once daily.

Lead-in Phase: Erlotinib + Entinostat 10 mg

Erlotinib 150 mg tablets, orally, daily plus entinostat 10 mg, tablets, orally, on Days 1 and 15 of each 28-day cycle until disease progression or intolerable toxicities for up to 6 cycles in the Lead-in Phase.

Group Type EXPERIMENTAL

Entinostat

Intervention Type DRUG

Entinostat tablets on Days 1 and 15 of a 28-day cycle.

Erlotinib

Intervention Type DRUG

Erlotinib 150 mg tablets once daily.

Double-blind Phase: Erlotinib + Entinostat 10 mg

Erlotinib 150 mg, tablets, orally, daily plus entinostat 10 mg, tablets, orally, on Day 1 and 15 of a 28-day cycle until disease progression or intolerable toxicities for up to 6 cycles in the Double-blind Phase.

Group Type EXPERIMENTAL

Entinostat

Intervention Type DRUG

Entinostat tablets on Days 1 and 15 of a 28-day cycle.

Erlotinib

Intervention Type DRUG

Erlotinib 150 mg tablets once daily.

Double-blind Phase: Erlotinib + Placebo

Erlotinib 150 mg, tablets, orally, daily plus placebo matching entinostat, tablets, orally, on Days 1 and 15 of each 28-day cycle until disease progression or intolerable toxicities for up to 6 cycles in the Double-blind Phase.

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Placebo-matching entinostat tablets on Days 1 and 15 of a 28-day cycle.

Erlotinib

Intervention Type DRUG

Erlotinib 150 mg tablets once daily.

Crossover Phase: Erlotinib + Entinostat 10 mg

Participants in the Double-blind Phase Erlotinib + Placebo arm who experienced disease progression crossed over to receive open-label erlotinib 150 mg, tablets, orally, daily plus entinostat 10 mg, tablets, orally, on Days 1 and 15 of each 28-day cycle until disease progression or intolerable toxicities.

Group Type EXPERIMENTAL

Entinostat

Intervention Type DRUG

Entinostat tablets on Days 1 and 15 of a 28-day cycle.

Erlotinib

Intervention Type DRUG

Erlotinib 150 mg tablets once daily.

Interventions

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Entinostat

Entinostat tablets on Days 1 and 15 of a 28-day cycle.

Intervention Type DRUG

Placebo

Placebo-matching entinostat tablets on Days 1 and 15 of a 28-day cycle.

Intervention Type DRUG

Erlotinib

Erlotinib 150 mg tablets once daily.

Intervention Type DRUG

Other Intervention Names

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SNDX-275 Tarceva

Eligibility Criteria

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Inclusion Criteria

* Cytologically or histologically confirmed NSCLC of stage IIIb or IV
* Received at least 1 but no more than 2 prior chemotherapy or chemoradiotherapy regimens for advanced NSCLC (that did not include erlotinib and valproic acid) and progressed based on radiologic evidence
* At least 1 measurable lesion by conventional or spiral computed tomography (CT) scan
* Eastern Cooperative Oncology Group (ECOG) performance score of 0, 1, or 2 and life expectancy of at least 6 months
* Paraffin-embedded tumor specimen available for correlative studies
* Male or female over 18 years of age
* Hemoglobin ≥ 9.0 g/dL; platelets ≥ 100 x 10\^9/L; absolute neutrophil count (ANC) ≥ 1.5 x 10\^9/L without the use of hematopoietic growth factors
* Bilirubin and creatinine less than 2 times the upper limit of normal for the institution
* Albumin ≥ 2.5 g/dL
* Aspartate aminotransferase (AST) and alanine aminotransferase (ALT) less than 3 times the upper limit of normal for the institution
* Prothrombin time less than 1.5 times the upper limit of normal for the institution
* Potassium, magnesium and phosphorus within the normal range for the institution (supplementation is permissible)
* Willing to use accepted and effective methods of contraception during the study (both men and women as appropriate) and for 3 months after the last dose of SNDX-275
* Patient or legally acceptable representative has granted written informed consent before any study-specific procedure (including special screening tests) are performed

Exclusion Criteria

* Prior stem cell transplant
* Clinical evidence of central nervous system (CNS) involvement
* Prior treatment with an histone deacetylase (HDAC) inhibitor or an epidermal growth factor receptor (EGFR) inhibitor
* Currently taking known inhibitors of CYPA4, including but not limited to atazanavir, clarithromycin, indinavir, itraconazole, nefazodone, nelfinavir, ritonavir, saquinavir, telithromycin, troleandomycin, ≥ 10 mg prednisone, and voriconazole
* Currently taking medication(s) on the prohibited medication list
* Prior exposure to SNDX-275
* Systemic chemotherapy, radiotherapy, or treatment with an investigational agent without recovery to at least grade 1 or baseline before study drug administration
* Daily treatment with ≥ 10 mg prednisone within 28 days before study drug administration
* Local or whole brain palliative radiotherapy within 14 days before study drug administration
* Currently active second malignancy, or any malignancy within the last 5 years other than cured basal or squamous cell skin carcinoma, cervical carcinoma in situ, carcinoma in situ of the bladder, or papillary thyroid cancer
* Inability to swallow oral medications or a gastrointestinal malabsorption condition
* Acute infection requiring intravenous (IV) antibiotics, antivirals, or antifungals within 14 days before study drug administration
* Known human immunodeficiency virus (HIV) infection, or active hepatitis B or C infection
* Another serious or uncontrolled medical condition within 90 days before study drug administration such as acute myocardial infarction, angina, ventricular arrhythmias, hypertension, diabetes mellitus, or renal or hepatic insufficiency
* Known hypersensitivity to benzamides
* Women who are currently pregnant or breast-feeding
* Patient currently is enrolled in (or completed within 28 days before study drug administration) another investigational drug study
* Patient has any kind of medical, psychiatric, or behavioral disorder that places the patient at increased risk for study participation or compromises the ability of the patient to give written informed consent and/or to comply with study procedures and requirements
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Syndax Pharmaceuticals

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Samir Witta, MD

Role: PRINCIPAL_INVESTIGATOR

Rocky Mountain Cancer Centers

Kartik Konduri, MD

Role: PRINCIPAL_INVESTIGATOR

Texas Oncology - Sammons Cancer Center

Robert Raju, MD

Role: PRINCIPAL_INVESTIGATOR

Dayton Oncology

Locations

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HOPE (Hematology Oncology Physicians & Extenders)

Tucson, Arizona, United States

Site Status

Rocky Mountain Cancer Center

Denver, Colorado, United States

Site Status

Advanced Medical Specialties

Miami, Florida, United States

Site Status

Ocala Oncology Center

Ocala, Florida, United States

Site Status

Cancer Centers of Florida

Ocoee, Florida, United States

Site Status

Hematology Oncology Associates of Illinois

Chicago, Illinois, United States

Site Status

Central Indiana Cancer Centers

Indianapolis, Indiana, United States

Site Status

Kansas City Cancer Centers

Overland Park, Kansas, United States

Site Status

Alliance Hematology Oncology

Westminster, Maryland, United States

Site Status

St Joseph Oncology

Saint Joseph, Missouri, United States

Site Status

The Center for Cancer Care & Research

St Louis, Missouri, United States

Site Status

Mahonig Valley Hematology Oncology Associates

Boardman, Ohio, United States

Site Status

Dayton Oncology & Hematology

Kettering, Ohio, United States

Site Status

Oncology Associates of Oregon

Eugene, Oregon, United States

Site Status

Texas Oncology

Amarillo, Texas, United States

Site Status

Texas Oncology

Austin, Texas, United States

Site Status

Texas Oncology

Bedford, Texas, United States

Site Status

Texas Oncology, Sammons Cancer Center

Dallas, Texas, United States

Site Status

Texas Oncology

Dallas, Texas, United States

Site Status

Texas Oncology

Fort Worth, Texas, United States

Site Status

Texas Oncology

Garland, Texas, United States

Site Status

Texas Oncology

Longview, Texas, United States

Site Status

Texas Oncology

Midland, Texas, United States

Site Status

Texas Oncology

Odessa, Texas, United States

Site Status

Texas Oncology

Tyler, Texas, United States

Site Status

Fairfax Northern Virginia Hematology-Oncology

Fairfax, Virginia, United States

Site Status

Virginia Oncology Associates

Norfolk, Virginia, United States

Site Status

Highline Medical Oncology

Burien, Washington, United States

Site Status

Cancer Care Northwest

Spokane, Washington, United States

Site Status

Yakima Valley Memorial Hospital/North Star Lodge

Yakima, Washington, United States

Site Status

Countries

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United States

Other Identifiers

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SNDX-275-0401

Identifier Type: -

Identifier Source: org_study_id

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