Trial Outcomes & Findings for A Phase 2, Dose Finding Study of PF-03187207 in Patients With Primary Open Angle Glaucoma or Ocular Hypertension. (NCT NCT00595101)

NCT ID: NCT00595101

Last Updated: 2020-09-14

Results Overview

Intraocular pressure (IOP) was measured using a Goldmann applanation tonometer. Diurnal IOP, defined as the mean IOP over the day based on values obtained at 8 AM, 10 AM, 1 PM, and 4 PM, was calculated for each visit. Both eyes were tested, with the right eye preceding the left eye. The operator initially set the dial at 10 mmHg, then looked through the slit lamp and adjusted the dial to take the reading, and then recorded the results. The procedure was repeated on the same eye twice consecutively. If the measurements were within 2 mmHg or less of each other, the mean of the 2 readings was recorded as the IOP at that time point. If the 2 readings were more than 2 mmHg of each other, a third (consecutive) reading was taken and the median (middle) IOP was recorded as the IOP at that time point.

Recruitment status

COMPLETED

Study phase

PHASE2

Target enrollment

117 participants

Primary outcome timeframe

Baseline, 28 days

Results posted on

2020-09-14

Participant Flow

Participant milestones

Participant milestones
Measure
PF-0318 0.006%
PF-0318 0.006% once daily in the evening
PF-0318 0.024%
PF-0318 0.024% once daily in the evening
PF-0318 0.04%
PF-0318 0.04% once daily in the evening
0.005% Latanoprost
0.005% latanoprost once daily in the evening
Overall Study
STARTED
29
29
29
30
Overall Study
COMPLETED
29
28
29
30
Overall Study
NOT COMPLETED
0
1
0
0

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

A Phase 2, Dose Finding Study of PF-03187207 in Patients With Primary Open Angle Glaucoma or Ocular Hypertension.

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
PF-0318 0.006%
n=29 Participants
PF-0318 0.006% once daily in the evening
PF-0318 0.024%
n=29 Participants
PF-0318 0.024% once daily in the evening
PF-0318 0.04%
n=29 Participants
PF-0318 0.04% once daily in the evening
0.005% Latanoprost
n=30 Participants
0.005% latanoprost once daily in the evening
Total
n=117 Participants
Total of all reporting groups
Age, Continuous
58.3 years
STANDARD_DEVIATION 12.2 • n=5 Participants
60.9 years
STANDARD_DEVIATION 18.0 • n=7 Participants
58.8 years
STANDARD_DEVIATION 15.1 • n=5 Participants
60.0 years
STANDARD_DEVIATION 17.3 • n=4 Participants
59.5 years
STANDARD_DEVIATION 15.7 • n=21 Participants
Sex: Female, Male
Female
13 Participants
n=5 Participants
12 Participants
n=7 Participants
18 Participants
n=5 Participants
16 Participants
n=4 Participants
59 Participants
n=21 Participants
Sex: Female, Male
Male
16 Participants
n=5 Participants
17 Participants
n=7 Participants
11 Participants
n=5 Participants
14 Participants
n=4 Participants
58 Participants
n=21 Participants

PRIMARY outcome

Timeframe: Baseline, 28 days

Population: The Per Protocol (PP) population consisted of all subjects in the intention to treat (ITT) population excluding those who made major protocol violations before completing the study. The PP population was considered as the primary analysis population of efficacy (primary and secondary endpoints) of the study.

Intraocular pressure (IOP) was measured using a Goldmann applanation tonometer. Diurnal IOP, defined as the mean IOP over the day based on values obtained at 8 AM, 10 AM, 1 PM, and 4 PM, was calculated for each visit. Both eyes were tested, with the right eye preceding the left eye. The operator initially set the dial at 10 mmHg, then looked through the slit lamp and adjusted the dial to take the reading, and then recorded the results. The procedure was repeated on the same eye twice consecutively. If the measurements were within 2 mmHg or less of each other, the mean of the 2 readings was recorded as the IOP at that time point. If the 2 readings were more than 2 mmHg of each other, a third (consecutive) reading was taken and the median (middle) IOP was recorded as the IOP at that time point.

Outcome measures

Outcome measures
Measure
PF-0318 0.006%
n=28 Participants
PF-0318 0.006% once daily in the evening
PF-0318 0.024%
n=27 Participants
PF-0318 0.024% once daily in the evening
PF-0318 0.04%
n=27 Participants
PF-0318 0.04% once daily in the evening
0.005% Latanoprost
n=30 Participants
0.005% latanoprost once daily in the evening
Change From Baseline Mean Diurnal Intraocular Pressure (IOP) in the Study Eye on Day 28
-5.12 mmHg (milimeters of mercury)
Standard Deviation 2.55
-5.94 mmHg (milimeters of mercury)
Standard Deviation 3.09
-5.02 mmHg (milimeters of mercury)
Standard Deviation 2.03
-5.25 mmHg (milimeters of mercury)
Standard Deviation 2.53

SECONDARY outcome

Timeframe: Baseline, Day 14, Day 28

Population: The Per Protocol (PP) population consisted of all subjects in the intention to treat (ITT) population excluding those who made major protocol violations before completing the study. The PP population was considered as the primary analysis population of efficacy (primary and secondary endpoints) of the study.

Intraocular pressure (IOP) was measured using a Goldmann applanation tonometer. Both eyes were tested, with the right eye preceding the left eye. The operator initially set the dial at 10 mmHg, then looked through the slit lamp and adjusted the dial to take the reading, and then recorded the results. The procedure was repeated on the same eye twice consecutively. If the measurements were within 2 mmHg or less of each other, the mean of the 2 readings was recorded as the IOP at that time point. If the 2 readings were more than 2 mmHg of each other, a third (consecutive) reading was taken and the median (middle) IOP was recorded as the IOP at that time point.

Outcome measures

Outcome measures
Measure
PF-0318 0.006%
n=28 Participants
PF-0318 0.006% once daily in the evening
PF-0318 0.024%
n=27 Participants
PF-0318 0.024% once daily in the evening
PF-0318 0.04%
n=27 Participants
PF-0318 0.04% once daily in the evening
0.005% Latanoprost
n=30 Participants
0.005% latanoprost once daily in the evening
Change From Baseline in Mean Intraocular Pressure (IOP) at Specific Time Points on Day 14 and Day 28
Day 28, 2pm
-4.57 mmHg (milimeters of mercury)
Standard Deviation 2.77
-5.28 mmHg (milimeters of mercury)
Standard Deviation 3.17
-4.85 mmHg (milimeters of mercury)
Standard Deviation 2.11
-5.27 mmHg (milimeters of mercury)
Standard Deviation 3.11
Change From Baseline in Mean Intraocular Pressure (IOP) at Specific Time Points on Day 14 and Day 28
Day 28, 5pm
-4.68 mmHg (milimeters of mercury)
Standard Deviation 2.47
-6.28 mmHg (milimeters of mercury)
Standard Deviation 3.56
-4.57 mmHg (milimeters of mercury)
Standard Deviation 2.53
-4.73 mmHg (milimeters of mercury)
Standard Deviation 2.93
Change From Baseline in Mean Intraocular Pressure (IOP) at Specific Time Points on Day 14 and Day 28
Day 14, 9am
-5.20 mmHg (milimeters of mercury)
Standard Deviation 2.97
-5.87 mmHg (milimeters of mercury)
Standard Deviation 3.21
-4.35 mmHg (milimeters of mercury)
Standard Deviation 2.76
-5.53 mmHg (milimeters of mercury)
Standard Deviation 2.53
Change From Baseline in Mean Intraocular Pressure (IOP) at Specific Time Points on Day 14 and Day 28
Day 28, 9am
-5.63 mmHg (milimeters of mercury)
Standard Deviation 3.29
-6.11 mmHg (milimeters of mercury)
Standard Deviation 3.82
-5.19 mmHg (milimeters of mercury)
Standard Deviation 2.71
-5.33 mmHg (milimeters of mercury)
Standard Deviation 2.66
Change From Baseline in Mean Intraocular Pressure (IOP) at Specific Time Points on Day 14 and Day 28
Day 28, 11am
-5.61 mmHg (milimeters of mercury)
Standard Deviation 3.20
-6.07 mmHg (milimeters of mercury)
Standard Deviation 3.31
-5.46 mmHg (milimeters of mercury)
Standard Deviation 2.56
-5.65 mmHg (milimeters of mercury)
Standard Deviation 2.80

SECONDARY outcome

Timeframe: Up to 28 days

Population: The Per Protocol (PP) population consisted of all subjects in the intention to treat (ITT) population excluding those who made major protocol violations before completing the study. The PP population was considered as the primary analysis population of efficacy (primary and secondary endpoints) of the study.

Percentage of participants with IOP of 18 mmHg or Lower, 16 mmHg or Lower, or 14 mmHg or Lower at Any Visit Through Day 28. Intraocular pressure (IOP) was measured using a Goldmann applanation tonometer. Both eyes were tested, with the right eye preceding the left eye. The operator initially set the dial at 10 mmHg, then looked through the slit lamp and adjusted the dial to take the reading, and then recorded the results. The procedure was repeated on the same eye twice consecutively. If the measurements were within 2 mmHg or less of each other, the mean of the 2 readings was recorded as the IOP at that time point. If the 2 readings were more than 2 mmHg of each other, a third (consecutive) reading was taken and the median (middle) IOP was recorded as the IOP at that time point.

Outcome measures

Outcome measures
Measure
PF-0318 0.006%
n=28 Participants
PF-0318 0.006% once daily in the evening
PF-0318 0.024%
n=27 Participants
PF-0318 0.024% once daily in the evening
PF-0318 0.04%
n=27 Participants
PF-0318 0.04% once daily in the evening
0.005% Latanoprost
n=30 Participants
0.005% latanoprost once daily in the evening
Target IOP
16 mmHg or lower
4 Participants
2 Participants
3 Participants
3 Participants
Target IOP
18 mmHg or lower
9 Participants
11 Participants
13 Participants
9 Participants
Target IOP
14 mmHg or lower
0 Participants
1 Participants
0 Participants
2 Participants

Adverse Events

PF-0318 0.006%

Serious events: 0 serious events
Other events: 2 other events
Deaths: 0 deaths

PF-0318 0.024%

Serious events: 0 serious events
Other events: 3 other events
Deaths: 0 deaths

PF-0318 0.04%

Serious events: 0 serious events
Other events: 5 other events
Deaths: 0 deaths

0.005% Latanoprost

Serious events: 0 serious events
Other events: 2 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
PF-0318 0.006%
n=29 participants at risk
PF-0318 0.006% once daily in the evening
PF-0318 0.024%
n=29 participants at risk
PF-0318 0.024% once daily in the evening
PF-0318 0.04%
n=29 participants at risk
PF-0318 0.04% once daily in the evening
0.005% Latanoprost
n=30 participants at risk
0.005% latanoprost once daily in the evening
Eye disorders
Conjunctival hyperaemia
0.00%
0/29 • 28 days
10.3%
3/29 • 28 days
0.00%
0/29 • 28 days
0.00%
0/30 • 28 days
Eye disorders
Ocular hyperaemia
3.4%
1/29 • 28 days
3.4%
1/29 • 28 days
6.9%
2/29 • 28 days
3.3%
1/30 • 28 days
Infections and infestations
Nasopharyngitis
3.4%
1/29 • 28 days
3.4%
1/29 • 28 days
10.3%
3/29 • 28 days
6.7%
2/30 • 28 days

Additional Information

Study Director

Bausch Health

Phone: 908-300-9920

Results disclosure agreements

  • Principal investigator is a sponsor employee Contact sponsor directly for details
  • Publication restrictions are in place

Restriction type: OTHER