Trial Outcomes & Findings for Study Evaluating Oral MOA-728 For The Treatment Of OIBD In Subjects With Chronic Non-Malignant Pain (NCT NCT00547586)

NCT ID: NCT00547586

Last Updated: 2020-08-20

Results Overview

Recruitment status

COMPLETED

Study phase

PHASE2

Target enrollment

122 participants

Primary outcome timeframe

6 hours

Results posted on

2020-08-20

Participant Flow

Participant milestones

Participant milestones
Measure
Placebo
placebo: placebo
150 mg
N-methylnaltrexone bromide (MOA-728): Oral
300 mg
N-methylnaltrexone bromide (MOA-728): Oral
450 mg
N-methylnaltrexone bromide (MOA-728): Oral
600 mg
N-methylnaltrexone bromide (MOA-728): Oral
Overall Study
STARTED
33
7
14
33
35
Overall Study
COMPLETED
28
6
13
27
32
Overall Study
NOT COMPLETED
5
1
1
6
3

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

Study Evaluating Oral MOA-728 For The Treatment Of OIBD In Subjects With Chronic Non-Malignant Pain

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Placebo
n=33 Participants
placebo: placebo
150 mg
n=7 Participants
N-methylnaltrexone bromide (MOA-728): Oral
300 mg
n=14 Participants
N-methylnaltrexone bromide (MOA-728): Oral
450 mg
n=33 Participants
N-methylnaltrexone bromide (MOA-728): Oral
600 mg
n=35 Participants
N-methylnaltrexone bromide (MOA-728): Oral
Total
n=122 Participants
Total of all reporting groups
Age, Continuous
48 years
STANDARD_DEVIATION 8.75 • n=5 Participants
48.43 years
STANDARD_DEVIATION 6.80 • n=7 Participants
52.43 years
STANDARD_DEVIATION 8.56 • n=5 Participants
51.21 years
STANDARD_DEVIATION 12.24 • n=4 Participants
49.51 years
STANDARD_DEVIATION 11.25 • n=21 Participants
49.84 years
STANDARD_DEVIATION 10.39 • n=10 Participants
Sex: Female, Male
Female
22 Participants
n=5 Participants
5 Participants
n=7 Participants
5 Participants
n=5 Participants
24 Participants
n=4 Participants
18 Participants
n=21 Participants
74 Participants
n=10 Participants
Sex: Female, Male
Male
11 Participants
n=5 Participants
2 Participants
n=7 Participants
9 Participants
n=5 Participants
9 Participants
n=4 Participants
17 Participants
n=21 Participants
48 Participants
n=10 Participants

PRIMARY outcome

Timeframe: 6 hours

Outcome measures

Outcome measures
Measure
Placebo
n=33 Participants
placebo: placebo
150 mg
n=7 Participants
N-methylnaltrexone bromide (MOA-728): Oral
300 mg
n=14 Participants
N-methylnaltrexone bromide (MOA-728): Oral
450 mg
n=33 Participants
N-methylnaltrexone bromide (MOA-728): Oral
600 mg
n=35 Participants
N-methylnaltrexone bromide (MOA-728): Oral
Percentage of Participants With a Spontaneous Bowel Movement (SBM) Within 1, 2, 3, 4, and 6 Hours of Treatment
Within 1 hour of 1st dose
0 Participants
0 Participants
0 Participants
7 Participants
2 Participants
Percentage of Participants With a Spontaneous Bowel Movement (SBM) Within 1, 2, 3, 4, and 6 Hours of Treatment
Within 2 hours of 1st dose
1 Participants
1 Participants
1 Participants
9 Participants
5 Participants
Percentage of Participants With a Spontaneous Bowel Movement (SBM) Within 1, 2, 3, 4, and 6 Hours of Treatment
Within 3 hours of 1st dose
3 Participants
1 Participants
2 Participants
13 Participants
9 Participants
Percentage of Participants With a Spontaneous Bowel Movement (SBM) Within 1, 2, 3, 4, and 6 Hours of Treatment
Within 4 hours of 1st dose
3 Participants
1 Participants
4 Participants
15 Participants
14 Participants
Percentage of Participants With a Spontaneous Bowel Movement (SBM) Within 1, 2, 3, 4, and 6 Hours of Treatment
Within 6 hours of 1st dose
6 Participants
1 Participants
4 Participants
15 Participants
17 Participants

Adverse Events

Placebo

Serious events: 0 serious events
Other events: 10 other events
Deaths: 15 deaths

150 mg

Serious events: 0 serious events
Other events: 3 other events
Deaths: 3 deaths

300 mg

Serious events: 0 serious events
Other events: 4 other events
Deaths: 4 deaths

450 mg

Serious events: 1 serious events
Other events: 9 other events
Deaths: 13 deaths

600 mg

Serious events: 3 serious events
Other events: 6 other events
Deaths: 18 deaths

Serious adverse events

Serious adverse events
Measure
Placebo
n=33 participants at risk
placebo: placebo
150 mg
n=7 participants at risk
N-methylnaltrexone bromide (MOA-728): Oral
300 mg
n=14 participants at risk
N-methylnaltrexone bromide (MOA-728): Oral
450 mg
n=33 participants at risk
N-methylnaltrexone bromide (MOA-728): Oral
600 mg
n=35 participants at risk
N-methylnaltrexone bromide (MOA-728): Oral
General disorders
Lymphedema
0.00%
0/33 • 6 weeks
0.00%
0/7 • 6 weeks
0.00%
0/14 • 6 weeks
0.00%
0/33 • 6 weeks
2.9%
1/35 • 6 weeks
General disorders
Pain
0.00%
0/33 • 6 weeks
0.00%
0/7 • 6 weeks
0.00%
0/14 • 6 weeks
0.00%
0/33 • 6 weeks
2.9%
1/35 • 6 weeks
Infections and infestations
Cellulitis staphyloccocal
0.00%
0/33 • 6 weeks
0.00%
0/7 • 6 weeks
0.00%
0/14 • 6 weeks
0.00%
0/33 • 6 weeks
2.9%
1/35 • 6 weeks
Infections and infestations
Bursitis infective
0.00%
0/33 • 6 weeks
0.00%
0/7 • 6 weeks
0.00%
0/14 • 6 weeks
0.00%
0/33 • 6 weeks
2.9%
1/35 • 6 weeks
Injury, poisoning and procedural complications
Overdose
0.00%
0/33 • 6 weeks
0.00%
0/7 • 6 weeks
0.00%
0/14 • 6 weeks
0.00%
0/33 • 6 weeks
2.9%
1/35 • 6 weeks
Gastrointestinal disorders
Small intestinal obstruction
0.00%
0/33 • 6 weeks
0.00%
0/7 • 6 weeks
0.00%
0/14 • 6 weeks
0.00%
0/33 • 6 weeks
2.9%
1/35 • 6 weeks
Injury, poisoning and procedural complications
Accidental overdose
0.00%
0/33 • 6 weeks
0.00%
0/7 • 6 weeks
0.00%
0/14 • 6 weeks
3.0%
1/33 • 6 weeks
0.00%
0/35 • 6 weeks

Other adverse events

Other adverse events
Measure
Placebo
n=33 participants at risk
placebo: placebo
150 mg
n=7 participants at risk
N-methylnaltrexone bromide (MOA-728): Oral
300 mg
n=14 participants at risk
N-methylnaltrexone bromide (MOA-728): Oral
450 mg
n=33 participants at risk
N-methylnaltrexone bromide (MOA-728): Oral
600 mg
n=35 participants at risk
N-methylnaltrexone bromide (MOA-728): Oral
Gastrointestinal disorders
Abdominal discomfort
0.00%
0/33 • 6 weeks
14.3%
1/7 • 6 weeks
0.00%
0/14 • 6 weeks
0.00%
0/33 • 6 weeks
0.00%
0/35 • 6 weeks
Gastrointestinal disorders
Abdominal distention
6.1%
2/33 • 6 weeks
0.00%
0/7 • 6 weeks
0.00%
0/14 • 6 weeks
6.1%
2/33 • 6 weeks
0.00%
0/35 • 6 weeks
Gastrointestinal disorders
Abdominal pain
0.00%
0/33 • 6 weeks
0.00%
0/7 • 6 weeks
14.3%
2/14 • 6 weeks
6.1%
2/33 • 6 weeks
2.9%
1/35 • 6 weeks
Gastrointestinal disorders
Diarrhea
0.00%
0/33 • 6 weeks
14.3%
1/7 • 6 weeks
0.00%
0/14 • 6 weeks
6.1%
2/33 • 6 weeks
5.7%
2/35 • 6 weeks
Gastrointestinal disorders
Flatulence
6.1%
2/33 • 6 weeks
0.00%
0/7 • 6 weeks
7.1%
1/14 • 6 weeks
0.00%
0/33 • 6 weeks
0.00%
0/35 • 6 weeks
Gastrointestinal disorders
Gastrointestinal motility disorder
0.00%
0/33 • 6 weeks
0.00%
0/7 • 6 weeks
7.1%
1/14 • 6 weeks
0.00%
0/33 • 6 weeks
0.00%
0/35 • 6 weeks
Gastrointestinal disorders
Nausea
9.1%
3/33 • 6 weeks
14.3%
1/7 • 6 weeks
7.1%
1/14 • 6 weeks
3.0%
1/33 • 6 weeks
2.9%
1/35 • 6 weeks
Gastrointestinal disorders
Vomiting
3.0%
1/33 • 6 weeks
0.00%
0/7 • 6 weeks
0.00%
0/14 • 6 weeks
6.1%
2/33 • 6 weeks
0.00%
0/35 • 6 weeks
Infections and infestations
Herpes zoster
0.00%
0/33 • 6 weeks
14.3%
1/7 • 6 weeks
0.00%
0/14 • 6 weeks
0.00%
0/33 • 6 weeks
0.00%
0/35 • 6 weeks
Infections and infestations
Influenza
6.1%
2/33 • 6 weeks
0.00%
0/7 • 6 weeks
0.00%
0/14 • 6 weeks
0.00%
0/33 • 6 weeks
2.9%
1/35 • 6 weeks
Infections and infestations
Urinary tract infection
3.0%
1/33 • 6 weeks
0.00%
0/7 • 6 weeks
7.1%
1/14 • 6 weeks
0.00%
0/33 • 6 weeks
2.9%
1/35 • 6 weeks
Injury, poisoning and procedural complications
Tooth fracture
0.00%
0/33 • 6 weeks
14.3%
1/7 • 6 weeks
0.00%
0/14 • 6 weeks
0.00%
0/33 • 6 weeks
0.00%
0/35 • 6 weeks
Musculoskeletal and connective tissue disorders
Bone pain
0.00%
0/33 • 6 weeks
14.3%
1/7 • 6 weeks
0.00%
0/14 • 6 weeks
0.00%
0/33 • 6 weeks
0.00%
0/35 • 6 weeks
Nervous system disorders
Headache
0.00%
0/33 • 6 weeks
0.00%
0/7 • 6 weeks
7.1%
1/14 • 6 weeks
0.00%
0/33 • 6 weeks
2.9%
1/35 • 6 weeks

Additional Information

Study Director

Bausch Health

Results disclosure agreements

  • Principal investigator is a sponsor employee Contact sponsor directly for details.
  • Publication restrictions are in place

Restriction type: OTHER