Vinorelbine in Treating Patients With Advanced Solid Tumors That Have Not Responded to Treatment and Liver Dysfunction

NCT ID: NCT00540982

Last Updated: 2025-07-02

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1/PHASE2

Total Enrollment

47 participants

Study Classification

INTERVENTIONAL

Study Start Date

1997-02-20

Study Completion Date

2010-05-20

Brief Summary

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RATIONALE: Drugs used in chemotherapy, such as vinorelbine, work in different ways to stop the growth of tumor cells, either by killing the cells or by stopping them from dividing.

PURPOSE: This pilot trial is studying the side effects and best dose of vinorelbine in treating patients with advanced solid tumors that have not responded to treatment and liver dysfunction.

Detailed Description

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OBJECTIVES:

* To correlate indocyanine green and lidocaine metabolism with vinorelbine ditartrate pharmacokinetics in patients with advanced, refractory solid tumors and varying degrees of liver dysfunction.
* To determine the pharmacokinetics of vinorelbine ditartrate in these patients.
* To test a plan of dose adjustment for vinorelbine ditartrate administration in these patients.

OUTLINE: Patients are stratified according to extent of clinical liver dysfunction (normal vs mild vs moderate vs severe).

Patients receive dose-adjusted vinorelbine ditartrate IV over 10 minutes once weekly in the absence of disease progression or unacceptable toxicity. Patients achieving an objective complete response receive 2 additional courses of study therapy.

Patients undergo blood sample collection periodically during study for pharmacokinetic and pharmacodynamic correlative studies. Blood is also collected after patients receive lidocaine IV push and indocyanine green (ICG) IV push. Samples are analyzed for whole blood and plasma concentrations of vinorelbine ditartrate and its metabolites by high performance liquid chromatography (15) or by liquid chromatography/tandem mass spectrometry assay. Samples are also analyzed for ICG clearance and lidocaine hydrochloride metabolic capacity by fluorescent polarization immunoassay.

After completion of study therapy, patients are followed periodically.

Conditions

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Lung Cancer Unspecified Adult Solid Tumor, Protocol Specific

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Normal Liver Function

Group Type EXPERIMENTAL

indocyanine green

Intervention Type DRUG

0.5 mg/kg will be administered by IV push to determine clearance

lidocaine

Intervention Type DRUG

1 mg/kg will be administered to determine metabolic capacity

vinorelbine ditartrate

Intervention Type DRUG

Varying doses ranging from 30 mg/m2 to 7.5 mg/m2 will be administered based upon liver function

high performance liquid chromatography

Intervention Type OTHER

Used to determine plasma concentrations of vinorelbine

intracellular fluorescence polarization analysis

Intervention Type OTHER

Used to determine concentration of lidocaine metabolic capacity

liquid chromatography

Intervention Type OTHER

Used to determine concentrations of vinorelbine and its metabolites

mass spectrometry

Intervention Type OTHER

Used to determine concentrations of vinorelbine and its metabolites

pharmacological study

Intervention Type OTHER

Determination of concentrations of vinorelbine and its metabolites

Mild Liver Dysfunction

Group Type EXPERIMENTAL

indocyanine green

Intervention Type DRUG

0.5 mg/kg will be administered by IV push to determine clearance

lidocaine

Intervention Type DRUG

1 mg/kg will be administered to determine metabolic capacity

vinorelbine ditartrate

Intervention Type DRUG

Varying doses ranging from 30 mg/m2 to 7.5 mg/m2 will be administered based upon liver function

high performance liquid chromatography

Intervention Type OTHER

Used to determine plasma concentrations of vinorelbine

intracellular fluorescence polarization analysis

Intervention Type OTHER

Used to determine concentration of lidocaine metabolic capacity

liquid chromatography

Intervention Type OTHER

Used to determine concentrations of vinorelbine and its metabolites

mass spectrometry

Intervention Type OTHER

Used to determine concentrations of vinorelbine and its metabolites

pharmacological study

Intervention Type OTHER

Determination of concentrations of vinorelbine and its metabolites

Moderate Liver Dysfunction

Group Type EXPERIMENTAL

indocyanine green

Intervention Type DRUG

0.5 mg/kg will be administered by IV push to determine clearance

lidocaine

Intervention Type DRUG

1 mg/kg will be administered to determine metabolic capacity

vinorelbine ditartrate

Intervention Type DRUG

Varying doses ranging from 30 mg/m2 to 7.5 mg/m2 will be administered based upon liver function

high performance liquid chromatography

Intervention Type OTHER

Used to determine plasma concentrations of vinorelbine

intracellular fluorescence polarization analysis

Intervention Type OTHER

Used to determine concentration of lidocaine metabolic capacity

liquid chromatography

Intervention Type OTHER

Used to determine concentrations of vinorelbine and its metabolites

mass spectrometry

Intervention Type OTHER

Used to determine concentrations of vinorelbine and its metabolites

pharmacological study

Intervention Type OTHER

Determination of concentrations of vinorelbine and its metabolites

Severe Liver Dysfunction

Group Type EXPERIMENTAL

indocyanine green

Intervention Type DRUG

0.5 mg/kg will be administered by IV push to determine clearance

lidocaine

Intervention Type DRUG

1 mg/kg will be administered to determine metabolic capacity

vinorelbine ditartrate

Intervention Type DRUG

Varying doses ranging from 30 mg/m2 to 7.5 mg/m2 will be administered based upon liver function

high performance liquid chromatography

Intervention Type OTHER

Used to determine plasma concentrations of vinorelbine

intracellular fluorescence polarization analysis

Intervention Type OTHER

Used to determine concentration of lidocaine metabolic capacity

liquid chromatography

Intervention Type OTHER

Used to determine concentrations of vinorelbine and its metabolites

mass spectrometry

Intervention Type OTHER

Used to determine concentrations of vinorelbine and its metabolites

pharmacological study

Intervention Type OTHER

Determination of concentrations of vinorelbine and its metabolites

Interventions

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indocyanine green

0.5 mg/kg will be administered by IV push to determine clearance

Intervention Type DRUG

lidocaine

1 mg/kg will be administered to determine metabolic capacity

Intervention Type DRUG

vinorelbine ditartrate

Varying doses ranging from 30 mg/m2 to 7.5 mg/m2 will be administered based upon liver function

Intervention Type DRUG

high performance liquid chromatography

Used to determine plasma concentrations of vinorelbine

Intervention Type OTHER

intracellular fluorescence polarization analysis

Used to determine concentration of lidocaine metabolic capacity

Intervention Type OTHER

liquid chromatography

Used to determine concentrations of vinorelbine and its metabolites

Intervention Type OTHER

mass spectrometry

Used to determine concentrations of vinorelbine and its metabolites

Intervention Type OTHER

pharmacological study

Determination of concentrations of vinorelbine and its metabolites

Intervention Type OTHER

Eligibility Criteria

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Inclusion Criteria

* Not pregnant or nursing
* Negative pregnancy test
* Fertile patients must use effective contraception
* No concurrent illness (e.g., cardiovascular, pulmonary, or central nervous system) that is poorly controlled or of such severity that the investigator deems unwise to enter the patient on protocol
* Must have ability to comply with study treatment and required tests
* Obstructive jaundice requires a drainage procedure prior to study treatment

PRIOR CONCURRENT THERAPY:

* See Disease Characteristics
* Recovered from prior therapy
* At least 3 weeks since prior chemotherapy (6 weeks for mitomycin or nitrosourea therapy)
* No prior radiotherapy to \> 30% of the bone marrow or more than standard adjuvant pelvic radiotherapy for rectal cancer
Minimum Eligible Age

18 Years

Maximum Eligible Age

120 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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National Cancer Institute (NCI)

NIH

Sponsor Role collaborator

City of Hope Medical Center

OTHER

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Joseph Chao

Role: STUDY_CHAIR

City of Hope Medical Center

Locations

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City of Hope Medical Center

Duarte, California, United States

Site Status

City of Hope Medical Group

Pasadena, California, United States

Site Status

Countries

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United States

Other Identifiers

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P30CA033572

Identifier Type: NIH

Identifier Source: secondary_id

View Link

CHNMC-96032

Identifier Type: -

Identifier Source: secondary_id

CDR0000567457

Identifier Type: REGISTRY

Identifier Source: secondary_id

96032

Identifier Type: -

Identifier Source: org_study_id

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