3 TPV/RTV Doses in Multiple ARV Experienced Patients - Tipranavir Dose Defining Study

NCT ID: NCT00275444

Last Updated: 2023-12-01

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

216 participants

Study Classification

INTERVENTIONAL

Study Start Date

2002-03-29

Brief Summary

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A dose defining study of the protease inhibitor tipranavir (TPV), boosted with low dose ritonavir (RTV). Three dose combinations of TPV/RTV are administered to multiple antiretroviral experienced patients and the dose that achieves the best efficacy and safety as determined by evaluation of 2, 8, and 24-week virologic response and adverse event and laboratory profile measures would be selected for further clinical study.

Detailed Description

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Conditions

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HIV Infections

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Interventions

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Tipranavir

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Signed informed consent prior to trial participation.
* Human immunodeficiency virus 1 (HIV-1) infected males or females \> 18 years of age.
* At least 3 months experience taking Nucleoside reverse transcriptase inhibitors (NRTIs), Non-nucleoside reverse transcriptase inhibitor (NNRTIs), and Protease inhibitors (PIs).
* Current PI-based Antiretroviral (ARV) medication regimen for at least 3 months prior to randomization, and at least 3 months experience taking at least one other PI-based regimen.
* HIV-1 viral load ≥1000 copies/mL at screening.
* Genotypic resistance report indicating one or more primary PI resistance mutation(s), including 30N, 46I/L, 48V, 50V, 82A/F/T, 84V or 90M.
* Availability of 2 or more non-PI ARV medications by genotypic resistance testing, i.e. 2 drugs tested as "no evidence of resistance" or "possible resistance".
* Acceptable screening laboratory values that indicate adequate baseline organ function.
* Laboratory values are considered to be acceptable if severity is no higher than Grade 3 Gamma glutamyl transferase (GGT), Grade 2 cholesterol or triglycerides, and no higher than Grade 1 for all other tests based on the "Division of Acquired Immune Deficiency Syndrome" of National Institute of Health, USA - DAIDS - Grading Scale. All laboratory values outside these limits are subject to approval by Boehringer Ingelheim (BI).

Exclusion Criteria

* ARV medication naïve.
* Only one or no available ARV medications as determined by genotypic resistance testing.
* Female subjects who:

* have a positive serum pregnancy test at screening or during the study;
* are breast feeding;
* are planning to become pregnant;
* are not willing to use two methods of contraception to include at least one barrier method (e.g. latex condom plus spermicidal jelly/foam).
* Any active opportunistic infection within 60 days before study entry.
* Active Hepatitis B (HCB) or Hepatitis C (HCV) disease defined as HBsAg positive or HCV RNA positive with Aspartate aminotransferase (AST)/Alanine aminotransferase (ALT) \> Grade 1.
* Prior tipranavir use.
* Use of investigational medications within 30 days before study entry or during the trial.Some expanded access drugs may be acceptable; must be approved by BI. Tenofovir, investigational at time of preparation of this protocol, is acceptable.
* Use of concomitant drugs which may significantly reduce plasma levels of the study medications.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Boehringer Ingelheim

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Boehringer Ingelheim Study Coordinator

Role: STUDY_CHAIR

Boehringer Ingelheim

Locations

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Boehringer Ingelheim Investigational Site

Phoenix, Arizona, United States

Site Status

Boehringer Ingelheim Investigational Site

Fountain Valley, California, United States

Site Status

Living Hope Clinical Trials, Inc.

Long Beach, California, United States

Site Status

Boehringer Ingelheim Investigational Site

Los Angeles, California, United States

Site Status

David Geffen School of Medicine at UCLA

Los Angeles, California, United States

Site Status

Vincent Lombardi Cancer Center

Washington D.C., District of Columbia, United States

Site Status

Therafirst Medical Center

Fort Lauderdale, Florida, United States

Site Status

1501 N.W. 9th Ave

Miami, Florida, United States

Site Status

Boehringer Ingelheim Investigational Site

Orlando, Florida, United States

Site Status

Boehringer Ingelheim Investigational Site

South Miami, Florida, United States

Site Status

Hillsborough County Health Dept.

Tampa, Florida, United States

Site Status

Boehringer Ingelheim Investigational Site

Vero Beach, Florida, United States

Site Status

Boehringer Ingelheim Investigational Site

Atlanta, Georgia, United States

Site Status

Atlanta VA Medical Center

Decatur, Georgia, United States

Site Status

Mercer University School of Medicine

Macon, Georgia, United States

Site Status

CORE Center

Chicago, Illinois, United States

Site Status

Rush-Presbytarian-St Luke's Medical Center

Chicago, Illinois, United States

Site Status

University of Louisville

Louisville, Kentucky, United States

Site Status

HIV Outpatient Program (H.O.P)

New Orleans, Louisiana, United States

Site Status

John's Hopkins University

Baltimore, Maryland, United States

Site Status

Boehringer Ingelheim Investigational Site

Boston, Massachusetts, United States

Site Status

Community Research Initiative of New England

Springfield, Massachusetts, United States

Site Status

University of Michigan Health System

Ann Arbor, Michigan, United States

Site Status

Boehringer Ingelheim Investigational Site

Kansas City, Missouri, United States

Site Status

Washington University

St Louis, Missouri, United States

Site Status

Boehringer Ingelheim Investigational Site

Las Vegas, Nevada, United States

Site Status

ID Care

Hillsborough, New Jersey, United States

Site Status

Boehringer Ingelheim Investigational Site

Santa Fe, New Mexico, United States

Site Status

Albany Medical College

Albany, New York, United States

Site Status

University of New York at Stony Brook

Stony Brook, New York, United States

Site Status

Duke University Medical Center

Durham, North Carolina, United States

Site Status

Boehringer Ingelheim Investigational Site

Huntersville, North Carolina, United States

Site Status

Wake Forest University Baptist Medical Center

Winston-Salem, North Carolina, United States

Site Status

Ohio State University Medical Center

Columbus, Ohio, United States

Site Status

Boehringer Ingelheim Investigational Site

Oklahoma City, Oklahoma, United States

Site Status

Boehringer Ingelheim Investigational Site

Columbia, South Carolina, United States

Site Status

Boehringer Ingelheim Investigational Site

Houston, Texas, United States

Site Status

Boehringer Ingelheim Investigational Site

Annandale, Virginia, United States

Site Status

Boehringer Ingelheim Investigational Site

Darlinghurst, New South Wales, Australia

Site Status

St. Vincent's Hospital

Darlinghurst, New South Wales, Australia

Site Status

Boehringer Ingelheim Investigational Site

Ottawa, Ontario, Canada

Site Status

Toronto General Hospital

Toronto, Ontario, Canada

Site Status

Montreal Chest Institute - McGill University Health Centre

Montreal, Quebec, Canada

Site Status

Hôpital de Bicêtre

Le Kremlin-Bicêtre, , France

Site Status

Hôpital de Chauliac

Montpellier, , France

Site Status

Hôpital Hôtel Dieu

Nantes, , France

Site Status

Hôpital Bichat Claude Bernard

Paris, , France

Site Status

Hôpital de la pitié Salpetrière

Paris, , France

Site Status

Hôpital Saint Louis

Paris, , France

Site Status

Epimed GmbH

Berlin, , Germany

Site Status

Klinik I für Innere Medizin der

Cologne, , Germany

Site Status

Klinikum der J.-W.-Goethe-Universität

Frankfurt am Main, , Germany

Site Status

Medizinische Poliklinik

München, , Germany

Site Status

Fondazione Centro S. Raffaele del Monte Tabor

Milan, , Italy

Site Status

IRCCS Policlinico San Matteo

Pavia, , Italy

Site Status

Academisch Medisch Centrum

Amsterdam, , Netherlands

Site Status

Erasmus Medical Centre

Rotterdam, , Netherlands

Site Status

Hospital Clínico y Provincial de Barcelona - HIV

Barcelona, , Spain

Site Status

Boehringer Ingelheim Investigational Site

Madrid, , Spain

Site Status

Hospital La Paz.

Madrid, , Spain

Site Status

Hospital Ramón y Cajal.

Madrid, , Spain

Site Status

4th Floor Research Office (St Stephens Centre)

London, , United Kingdom

Site Status

Countries

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United States Australia Canada France Germany Italy Netherlands Spain United Kingdom

Other Identifiers

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1182.52

Identifier Type: -

Identifier Source: org_study_id