NES Gel-1, To Evaluate Nestorone Gel in Combination With Testosterone Gel

NCT ID: NCT00229593

Last Updated: 2014-12-04

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

140 participants

Study Classification

INTERVENTIONAL

Study Start Date

2005-09-30

Study Completion Date

2007-01-31

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

The purpose of this study is to determine the usefulness of two transdermal gels to be used in the future development for a male contraceptive.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

The success of hormonal male contraception depends on the near complete suppression of spermatogenesis without producing any untoward effects on libido or other androgen-dependent functions or any other adverse events. The treatment with androgen alone has geen shown to be highly effective in Asian men but less effective in non-Asian men in clinical trials. To increase the efficacy of androgen alone treatment on spermatogenesis, combined regimens of a progestin and an androgen have shown promising results. The steady-state delivery of a progestin and an androgen by transdermal gel application would be a user-friendly delivery method as compared to injectable or implant approaches. Nestorone (NES) is a synthetic progestin that does not have any androgenic and estrogenic activity and is not expected to have some of the undesirable side effects of other drugs.

We propose to evaluate whether NES gel alone or in combination with T gel applied transdermally will result in more effective suppression of gonadotropins than NES or T gel applied alone in healthy men. Fifty healthy male subjects, age 18-50 will be enrolled at each center (2 sites).

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Contraception

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

DIAGNOSTIC

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

1

100 mg Testosterone gel daily for 3 weeks

Group Type ACTIVE_COMPARATOR

Testosterone Gel

Intervention Type DRUG

100 mg Testosterone gel daily for 3 weeks

2

2 mg Nestorone gel daily for 3 weeks

Group Type ACTIVE_COMPARATOR

Nestorone gel

Intervention Type DRUG

2 to 8 mg Nestorone gel daily for 3 weeks depending on treatment group assignment

3

4 mg Nestorone gel daily for 3 weeks

Group Type ACTIVE_COMPARATOR

Nestorone gel

Intervention Type DRUG

2 to 8 mg Nestorone gel daily for 3 weeks depending on treatment group assignment

4

100 mg Testosterone gel + 2 mg Nestorone gel

Group Type ACTIVE_COMPARATOR

Nestorone gel

Intervention Type DRUG

2 to 8 mg Nestorone gel daily for 3 weeks depending on treatment group assignment

Testosterone Gel

Intervention Type DRUG

100 mg Testosterone gel daily for 3 weeks

5

100 mg Testosterone gel + 4 mg Nestorone gel

Group Type ACTIVE_COMPARATOR

Nestorone gel

Intervention Type DRUG

2 to 8 mg Nestorone gel daily for 3 weeks depending on treatment group assignment

Testosterone Gel

Intervention Type DRUG

100 mg Testosterone gel daily for 3 weeks

6

100 mg Testosterone Gel + 6 mg Nestorone Gel daily for 3 weeks

Group Type ACTIVE_COMPARATOR

Nestorone gel

Intervention Type DRUG

2 to 8 mg Nestorone gel daily for 3 weeks depending on treatment group assignment

Testosterone Gel

Intervention Type DRUG

100 mg Testosterone gel daily for 3 weeks

7

100 mg Testosterone Gel + 8 mg Nestorone gel daily for 3 weeks

Group Type ACTIVE_COMPARATOR

Nestorone gel

Intervention Type DRUG

2 to 8 mg Nestorone gel daily for 3 weeks depending on treatment group assignment

Testosterone Gel

Intervention Type DRUG

100 mg Testosterone gel daily for 3 weeks

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

Nestorone gel

2 to 8 mg Nestorone gel daily for 3 weeks depending on treatment group assignment

Intervention Type DRUG

Testosterone Gel

100 mg Testosterone gel daily for 3 weeks

Intervention Type DRUG

Other Intervention Names

Discover alternative or legacy names that may be used to describe the listed interventions across different sources.

Testim

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Healthy men
* Aged 18-50 years
* With normal clinical chemistry, serum levels of testosterone, PSA, gonadotropins within normal limits, and sperm concentration greater than 20 million/mL
* Subject or his partner willing to use a recognized effective method of contraception

Exclusion Criteria

* Men not living in area of clinics
* Clinically significant abnormal findings at screening
* Elevated PSA greater than 4
* Partners who are pregnant
* Abnormal laboratory values, liver or kidney dysfunction
* Sperm counts below 20 million/mL.
* Use of androgens or body building substances within 6 months of enrollment,
* Blood pressure greater than 140/90, history of hypertension, including hypertension controlled with treatment
* History of primary testicular disease or disorder of the hypothalamic-pituitary axis
* Hypersensitivity of progestins
* History of venous thromboembolism
* Benign or malignant liver tumors
* Active liver disease, history of reproductive dysfunction including vasectomy or infertility
* History of active or chronic cardiac, renal, hepatic or prostatic disease
* Diabetes mellitus or morbid obesity (body weight greater than 120% of ideal body weight)
* Known or suspected alcoholism or drug abuse
* Known dermatitis or severe skin disorder

Men desiring fertility within 6 months or participating in competitive sports where drug screening for prohibited substances (including anabolic steroids) is routine will be advised of the relative and temporary hazards that participating in this study may have for their fertility or sporting status.
Minimum Eligible Age

18 Years

Maximum Eligible Age

50 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

Yes

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Eunice Kennedy Shriver National Institute of Child Health and Human Development (NICHD)

NIH

Sponsor Role collaborator

University of Washington

OTHER

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

William Bremner

Study Principal Investigator

Responsibility Role PRINCIPAL_INVESTIGATOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

William J Bremner, MD, PhD

Role: PRINCIPAL_INVESTIGATOR

University of Washington

Christina Wang, MD

Role: PRINCIPAL_INVESTIGATOR

University of California, Los Angeles

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

Harbor-UCLA Medical Center

Torrance, California, United States

Site Status

University of Washington Medical Center

Seattle, Washington, United States

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States

References

Explore related publications, articles, or registry entries linked to this study.

Anawalt BD, Bebb RA, Bremner WJ, Matsumoto AM. A lower dosage levonorgestrel and testosterone combination effectively suppresses spermatogenesis and circulating gonadotropin levels with fewer metabolic effects than higher dosage combinations. J Androl. 1999 May-Jun;20(3):407-14.

Reference Type BACKGROUND
PMID: 10386821 (View on PubMed)

Anderson RA, Kinniburgh D, Baird DT. Suppression of spermatogenesis by etonogestrel implants with depot testosterone: potential for long-acting male contraception. J Clin Endocrinol Metab. 2002 Aug;87(8):3640-9. doi: 10.1210/jcem.87.8.8773.

Reference Type BACKGROUND
PMID: 12161488 (View on PubMed)

Bebb RA, Anawalt BD, Christensen RB, Paulsen CA, Bremner WJ, Matsumoto AM. Combined administration of levonorgestrel and testosterone induces more rapid and effective suppression of spermatogenesis than testosterone alone: a promising male contraceptive approach. J Clin Endocrinol Metab. 1996 Feb;81(2):757-62. doi: 10.1210/jcem.81.2.8636300.

Reference Type BACKGROUND
PMID: 8636300 (View on PubMed)

Brache V, Massai R, Mishell DR, Moo-Young AJ, Alvarez F, Salvatierra AM, Cochon L, Croxatto H, Robbins A, Faundes A. Ovarian function during use of Nestorone(R) subdermal implants. Contraception. 2000 Mar;61(3):199-204. doi: 10.1016/s0010-7824(00)00092-5.

Reference Type BACKGROUND
PMID: 10827334 (View on PubMed)

Cummings DE, Bremner WJ. Prospects for new hormonal male contraceptives. Endocrinol Metab Clin North Am. 1994 Dec;23(4):893-922.

Reference Type BACKGROUND
PMID: 7705326 (View on PubMed)

Diaz S, Schiappacasse V, Pavez M, Zepeda A, Moo-Young AJ, Brandeis A, Lahteenmaki P, Croxatto HB. Clinical trial with Nestorone subdermal contraceptive implants. Contraception. 1995 Jan;51(1):33-8. doi: 10.1016/0010-7824(94)00006-i.

Reference Type BACKGROUND
PMID: 7750282 (View on PubMed)

Gonzalo IT, Swerdloff RS, Nelson AL, Clevenger B, Garcia R, Berman N, Wang C. Levonorgestrel implants (Norplant II) for male contraception clinical trials: combination with transdermal and injectable testosterone. J Clin Endocrinol Metab. 2002 Aug;87(8):3562-72. doi: 10.1210/jcem.87.8.8710.

Reference Type BACKGROUND
PMID: 12161475 (View on PubMed)

Haukkamaa M, Laurikka-Routti M, Heikinheimo O, Moo-Young A. Contraception with subdermal implants releasing the progestin ST-1435: a dose-finding study. Contraception. 1992 Jan;45(1):49-55. doi: 10.1016/0010-7824(92)90140-o.

Reference Type BACKGROUND
PMID: 1591921 (View on PubMed)

Handelsman DJ, Conway AJ, Howe CJ, Turner L, Mackey MA. Establishing the minimum effective dose and additive effects of depot progestin in suppression of human spermatogenesis by a testosterone depot. J Clin Endocrinol Metab. 1996 Nov;81(11):4113-21. doi: 10.1210/jcem.81.11.8923869.

Reference Type BACKGROUND
PMID: 8923869 (View on PubMed)

Kamischke A, Heuermann T, Kruger K, von Eckardstein S, Schellschmidt I, Rubig A, Nieschlag E. An effective hormonal male contraceptive using testosterone undecanoate with oral or injectable norethisterone preparations. J Clin Endocrinol Metab. 2002 Feb;87(2):530-9. doi: 10.1210/jcem.87.2.8218.

Reference Type BACKGROUND
PMID: 11836281 (View on PubMed)

Kamischke A, Venherm S, Ploger D, von Eckardstein S, Nieschlag E. Intramuscular testosterone undecanoate and norethisterone enanthate in a clinical trial for male contraception. J Clin Endocrinol Metab. 2001 Jan;86(1):303-9. doi: 10.1210/jcem.86.1.7057.

Reference Type BACKGROUND
PMID: 11232016 (View on PubMed)

Mahabadi V, Amory JK, Swerdloff RS, Bremner WJ, Page ST, Sitruk-Ware R, Christensen PD, Kumar N, Tsong YY, Blithe D, Wang C. Combined transdermal testosterone gel and the progestin nestorone suppresses serum gonadotropins in men. J Clin Endocrinol Metab. 2009 Jul;94(7):2313-20. doi: 10.1210/jc.2008-2604. Epub 2009 Apr 14.

Reference Type RESULT
PMID: 19366848 (View on PubMed)

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

HHSN27500002;

Identifier Type: -

Identifier Source: secondary_id

04-3792-D 02

Identifier Type: OTHER

Identifier Source: secondary_id

26852-D

Identifier Type: -

Identifier Source: org_study_id