Study Evaluating SKI-606 (Bosutinib) In Advanced Malignant Solid Tumors

NCT ID: NCT00195260

Last Updated: 2013-02-11

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

151 participants

Study Classification

INTERVENTIONAL

Study Start Date

2004-10-31

Study Completion Date

2007-11-30

Brief Summary

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To evaluate the safety and tolerability of oral SKI-606 (bosutinib) administered on a daily schedule to subjects with advanced malignant solid tumors and to define a maximum tolerated dose (MTD) in this subject population.

Detailed Description

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Conditions

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Neoplasms

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Dose escalation

Dose finding study of monotherapy bosutinib in patients with advanced solid tumors.

Group Type EXPERIMENTAL

bosutinib

Intervention Type DRUG

Dose levels evaluated 50mg, 100mg, 200mg, 300mg, 400mg, 500mg and 600mg. 500mg was identified as MTD, however due to GI toxicities at that dose, 400mg was selected as the RP2D. Drug was administered as long as tolerable and disease under study did not worsen.

Colorectal Cancer

Enroll 30 patients at RP2D to further evaluate safety and efficacy in subgroup population.

Group Type EXPERIMENTAL

bosutinib

Intervention Type DRUG

400mg QD bosutinib, as long as tolerated and disease under study does not worsen.

Pancreatic Cancer

Enroll 30 patients at RP2D to further evaluate safety and efficacy in subgroup population.

Group Type EXPERIMENTAL

bosutinib

Intervention Type DRUG

400mg QD bosutinib, as long as tolerated and disease under study does not worsen.

Non-Small Cell Lung Cancer (NSCLC)

Enroll 30 patients at RP2D to further evaluate safety and efficacy in subgroup population.

Group Type EXPERIMENTAL

bosutinib

Intervention Type DRUG

400mg QD bosutinib, as long as tolerated and disease under study does not worsen.

Interventions

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bosutinib

Dose levels evaluated 50mg, 100mg, 200mg, 300mg, 400mg, 500mg and 600mg. 500mg was identified as MTD, however due to GI toxicities at that dose, 400mg was selected as the RP2D. Drug was administered as long as tolerable and disease under study did not worsen.

Intervention Type DRUG

bosutinib

400mg QD bosutinib, as long as tolerated and disease under study does not worsen.

Intervention Type DRUG

bosutinib

400mg QD bosutinib, as long as tolerated and disease under study does not worsen.

Intervention Type DRUG

bosutinib

400mg QD bosutinib, as long as tolerated and disease under study does not worsen.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Advanced or recurrent solid malignancy confirmed histologically or cytologically for which no effective therapy is available.
* Eastern Cooperative Oncology Group (ECOG) performance status of 0 - 1.
* Measurable disease as outlined by the modified Response Evaluation Criteria in Solid Tumors (RECIST) criteria.
* Other inclusion applies.

Exclusion Criteria

* Use of any systemic antitumor agents or any investigational agent within 28 days before the first dose of test article is administered.
* Prior exposure to SKI-606 or any other Src-kinase inhibitor, major surgery or radiotherapy within 14 days before the first dose of test article (recovery from previous surgery should be complete before day 1).
* Active central nervous system (CNS) metastases, as indicated by clinical symptoms, cerebral edema, requirement for corticosteroids and/or progressive growth (Treated CNS metastases must be stable for \>= 2 weeks before day 1).
* Other exclusion applies.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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Pfizer Investigational Site

Birmington, Alabama, United States

Site Status

Pfizer Investigational Site

Scottsdale, Arizona, United States

Site Status

Pfizer Investigational Site

Los Angeles, California, United States

Site Status

Pfizer Investigational Site

Tampa, Florida, United States

Site Status

Pfizer Investigational Site

Atlanta, Georgia, United States

Site Status

Pfizer Investigational Site

Indianpolis, Indiana, United States

Site Status

Pfizer Investigational Site

Baltimore, Maryland, United States

Site Status

Pfizer Investigational Site

Detroit, Michigan, United States

Site Status

Pfizer Investigational Site

Lansing, Michigan, United States

Site Status

Pfizer Investigational Site

New York, New York, United States

Site Status

Pfizer Investigational Site

New York, New York, United States

Site Status

Pfizer Investigational Site

Charlotte, North Carolina, United States

Site Status

Pfizer Investigational Site

Charlotte, North Carolina, United States

Site Status

Pfizer Investigational Site

UNC Chapel Hill, North Carolina, United States

Site Status

Pfizer Investigational Site

UNC Chapel Hill, North Carolina, United States

Site Status

Pfizer Investigational Site

Cleveland, Ohio, United States

Site Status

Pfizer Investigational Site

San Antonio, Texas, United States

Site Status

Pfizer Investigational Site

Tyler, Texas, United States

Site Status

Pfizer Investigational Site

Seattle, Washington, United States

Site Status

Countries

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United States

References

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Hsyu PH, Mould DR, Abbas R, Amantea M. Population pharmacokinetic and pharmacodynamic analysis of bosutinib. Drug Metab Pharmacokinet. 2014;29(6):441-8. doi: 10.2133/dmpk.DMPK-13-RG-126. Epub 2014 Jun 10.

Reference Type DERIVED
PMID: 24919837 (View on PubMed)

Other Identifiers

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B1871012

Identifier Type: -

Identifier Source: secondary_id

3160A1-100

Identifier Type: -

Identifier Source: org_study_id

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