Trial Outcomes & Findings for A Study With TMC125 in Human Immunodeficiency Virus (HIV) Type 1 Infected Patients, Who Were Treated With TMC125 Arm in a Sponsor-Selected TMC125 Study (NCT NCT00128830)

NCT ID: NCT00128830

Last Updated: 2013-06-20

Results Overview

Number of participants who reported at least 1 of the adverse events.

Recruitment status

COMPLETED

Study phase

PHASE2

Target enrollment

211 participants

Primary outcome timeframe

Up to 3 years

Results posted on

2013-06-20

Participant Flow

In this study, 211 participants were enrolled in 12 different countries. The majority of participants (49%) were enrolled in the United States.

In total, 211 participants (93 who rolled over from the etravirine arm of study TMC125-C203 (NCT00412646), 85 who rolled over from the etravirine arm of study TMC125-C223 (NCT00081978), 29 who rolled over from study TMC125-C211 (NCT00111280) and 4 who rolled over from study TMC125-C209) received treatment with etravirine.

Participant milestones

Participant milestones
Measure
Etravirine
800 mg twice daily (formulation TF035), and after formulation switch, 200 mg twice daily (formulation F060)
Overall Study
STARTED
211
Overall Study
COMPLETED
139
Overall Study
NOT COMPLETED
72

Reasons for withdrawal

Reasons for withdrawal
Measure
Etravirine
800 mg twice daily (formulation TF035), and after formulation switch, 200 mg twice daily (formulation F060)
Overall Study
Adverse Event
10
Overall Study
Withdrawal by Subject
14
Overall Study
Lost to Follow-up
4
Overall Study
Reached a virologic endpoint
29
Overall Study
Non-compliant
4
Overall Study
Discontinued or ineligible for study
2
Overall Study
Other
9

Baseline Characteristics

A Study With TMC125 in Human Immunodeficiency Virus (HIV) Type 1 Infected Patients, Who Were Treated With TMC125 Arm in a Sponsor-Selected TMC125 Study

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Etravirine
n=211 Participants
800 mg twice daily (formulation TF035), and after formulation switch, 200 mg twice daily (formulation F060)
Age Continuous
46.0 years
FULL_RANGE 7.56 • n=5 Participants
Sex: Female, Male
Female
21 Participants
n=5 Participants
Sex: Female, Male
Male
190 Participants
n=5 Participants
Race/Ethnicity, Customized
Asian
1 Participants
n=5 Participants
Race/Ethnicity, Customized
Black or African American
24 Participants
n=5 Participants
Race/Ethnicity, Customized
White
164 Participants
n=5 Participants
Race/Ethnicity, Customized
Hispanic
16 Participants
n=5 Participants
Race/Ethnicity, Customized
Other
6 Participants
n=5 Participants

PRIMARY outcome

Timeframe: Up to 3 years

Population: Intent-to-treat population: Participants who received at least 1 dose of study medication were included

Number of participants who reported at least 1 of the adverse events.

Outcome measures

Outcome measures
Measure
Viral Load More Than or Equal to 50 Copies/mL
n=211 Participants
Viral load more than or equal to 50 copies/mL at TMC125-C229 Baseline
Viral Load Less Than 50 Copies/mL
Viral load less than 50 copies/mL at TMC125-C229 Baseline
Number of Participants With Adverse Events
195 Participants

SECONDARY outcome

Timeframe: Week 48

Population: Intent-to-treat participants who received at least one dose of study medication with evaluable data at Week 48

Number of participants who had viral load more than or equal to 50 copies/mL and less than 50 copies/mL at TMC125-C229 baseline and who achieved virologic response (ie, viral load less than 50 copies/mL) at Week 48. The last visit of the TMC125 feeder study (TMC125-C203 \[NCT00412646\], TMC125-C223 \[NCT00081978\], TMC125 C211 \[NCT00111280\] or TMC125-C209 feeder studies) was considered to be the TMC125-C229 baseline.

Outcome measures

Outcome measures
Measure
Viral Load More Than or Equal to 50 Copies/mL
n=80 Participants
Viral load more than or equal to 50 copies/mL at TMC125-C229 Baseline
Viral Load Less Than 50 Copies/mL
n=93 Participants
Viral load less than 50 copies/mL at TMC125-C229 Baseline
Number of Participants Who Achieved Virologic Response (ie, Viral Load Less Than 50 Copies/mL) at Week 48
22 Participants
80 Participants

SECONDARY outcome

Timeframe: Week 96

Population: Intent-to-treat participants who received at least one dose of study medication with evaluable data at Week 96

Number of participants who had viral load more than or equal to 50 copies/mL and less than 50 copies/mL at TMC125-C229 baseline and who achieved virologic response (ie, viral load less than 50 copies/mL) at Week 96. The last visit of the TMC125 feeder study (TMC125-C203 \[NCT00412646\], TMC125-C223 \[NCT00081978\], TMC125 C211 \[NCT00111280\] or TMC125-C209 feeder studies) was considered to be the TMC125-C229 baseline.

Outcome measures

Outcome measures
Measure
Viral Load More Than or Equal to 50 Copies/mL
n=62 Participants
Viral load more than or equal to 50 copies/mL at TMC125-C229 Baseline
Viral Load Less Than 50 Copies/mL
n=83 Participants
Viral load less than 50 copies/mL at TMC125-C229 Baseline
Number of Participants Who Achieved Virologic Response (ie, Viral Load Less Than 50 Copies/mL) at Week 96
28 Participants
72 Participants

SECONDARY outcome

Timeframe: Week 96

Population: Intent-to-treat participants who received at least one dose of study medication with evaluable data at Week 96

Baseline considered for this outcome is the baseline in the respective TMC125-C229 feeder study (TMC125-C203 \[NCT00412646\], TMC125-C223 \[NCT00081978\], TMC125 C211 \[NCT00111280\] or TMC125-C209 feeder studies).

Outcome measures

Outcome measures
Measure
Viral Load More Than or Equal to 50 Copies/mL
n=181 Participants
Viral load more than or equal to 50 copies/mL at TMC125-C229 Baseline
Viral Load Less Than 50 Copies/mL
Viral load less than 50 copies/mL at TMC125-C229 Baseline
Number of Participants Who Achieved Virologic Response (ie, Viral Load Less Than 50 Copies/mL; Less Than 400 Copies/mL; and Greater Than or Equal to 1 Log 10 Decrease From Baseline) at Week 96
Viral load (VL) less than 50 copies/mL
105 Participants
Number of Participants Who Achieved Virologic Response (ie, Viral Load Less Than 50 Copies/mL; Less Than 400 Copies/mL; and Greater Than or Equal to 1 Log 10 Decrease From Baseline) at Week 96
Viral load less than 400 copies/mL
124 Participants
Number of Participants Who Achieved Virologic Response (ie, Viral Load Less Than 50 Copies/mL; Less Than 400 Copies/mL; and Greater Than or Equal to 1 Log 10 Decrease From Baseline) at Week 96
Viral load more than or equal to 1log10
132 Participants

SECONDARY outcome

Timeframe: Week 192

Population: Intent-to-treat participants who received at least one dose of study medication with evaluable data at Week 192

Baseline considered for this outcome is the baseline in the respective TMC125-C229 feeder study (TMC125-C203 \[NCT00412646\], TMC125-C223 \[NCT00081978\], TMC125 C211 \[NCT00111280\] or TMC125-C209 feeder studies).

Outcome measures

Outcome measures
Measure
Viral Load More Than or Equal to 50 Copies/mL
n=98 Participants
Viral load more than or equal to 50 copies/mL at TMC125-C229 Baseline
Viral Load Less Than 50 Copies/mL
Viral load less than 50 copies/mL at TMC125-C229 Baseline
Number of Participants Who Achieved Virologic Response (ie, Viral Load Less Than 50 Copies/mL; Viral Load Less Than 400 Copies/mL; and Greater Than or Equal to 1 log10 Decrease From Baseline) at Week 192
Viral load (VL) less than 50 copies/mL
69 Participants
Number of Participants Who Achieved Virologic Response (ie, Viral Load Less Than 50 Copies/mL; Viral Load Less Than 400 Copies/mL; and Greater Than or Equal to 1 log10 Decrease From Baseline) at Week 192
VL less than 400 copies/mL
81 Participants
Number of Participants Who Achieved Virologic Response (ie, Viral Load Less Than 50 Copies/mL; Viral Load Less Than 400 Copies/mL; and Greater Than or Equal to 1 log10 Decrease From Baseline) at Week 192
VL greater than or equal to 1log10
83 Participants

SECONDARY outcome

Timeframe: Week 48

Population: Intent-to-treat participants who received at least one dose of study medication with evaluable data at Week 48

The last visit of the TMC125 feeder study (TMC125-C203 \[NCT00412646\], TMC125-C223 \[NCT00081978\], TMC125 C211 \[NCT00111280\] or TMC125-C209 feeder studies) was considered to be the TMC125-C229 baseline.

Outcome measures

Outcome measures
Measure
Viral Load More Than or Equal to 50 Copies/mL
n=172 Participants
Viral load more than or equal to 50 copies/mL at TMC125-C229 Baseline
Viral Load Less Than 50 Copies/mL
Viral load less than 50 copies/mL at TMC125-C229 Baseline
Median Change From TMC125-C229 Basline in Cluster of Differentiation 4 (CD4+) Cell Count at Week 48
21.50 x 100000 cells/L
Interval -422.0 to 1119.0

SECONDARY outcome

Timeframe: Week 96

Population: Intent-to-treat participants who received at least one dose of study medication with evaluable data at Week 96

The last visit of the TMC125 feeder study (TMC125-C203 \[NCT00412646\], TMC125-C223 \[NCT00081978\], TMC125 C211 \[NCT00111280\] or TMC125-C209 feeder studies) was considered to be the TMC125-C229 baseline.

Outcome measures

Outcome measures
Measure
Viral Load More Than or Equal to 50 Copies/mL
n=142 Participants
Viral load more than or equal to 50 copies/mL at TMC125-C229 Baseline
Viral Load Less Than 50 Copies/mL
Viral load less than 50 copies/mL at TMC125-C229 Baseline
Median Change From TMC125-C229 Baseline in Cluster of Differentiation 4 (CD4+) Cell Count at Week 96
18.50 x 1000000 cells/L
Interval -460.0 to 391.0

SECONDARY outcome

Timeframe: Week 96

Population: Intent-to-treat participants who received at least one dose of study medication with evaluable data at Week 96

Baseline considered for this outcome is the baseline in the respective TMC125-C229 feeder study (TMC125-C203 \[NCT00412646\], TMC125-C223 \[NCT00081978\], TMC125 C211 \[NCT00111280\] or TMC125-C209 feeder studies).

Outcome measures

Outcome measures
Measure
Viral Load More Than or Equal to 50 Copies/mL
n=181 Participants
Viral load more than or equal to 50 copies/mL at TMC125-C229 Baseline
Viral Load Less Than 50 Copies/mL
Viral load less than 50 copies/mL at TMC125-C229 Baseline
Median Change in Cluster of Differentiation 4 (CD4+) Cell Count From Baseline in TMC125-C229 Feeder Study at Week 96
120.00 x 1000000 cells/mL
Interval -393.0 to 1590.0

SECONDARY outcome

Timeframe: Week 192

Population: Intent-to-treat participants who received at least one dose of study medication with evaluable data at Week 192

Baseline considered for this outcome is the baseline in the respective TMC125-C229 feeder study (TMC125-C203 \[NCT00412646\], TMC125-C223 \[NCT00081978\], TMC125 C211 \[NCT00111280\] or TMC125-C209 feeder studies).

Outcome measures

Outcome measures
Measure
Viral Load More Than or Equal to 50 Copies/mL
n=96 Participants
Viral load more than or equal to 50 copies/mL at TMC125-C229 Baseline
Viral Load Less Than 50 Copies/mL
Viral load less than 50 copies/mL at TMC125-C229 Baseline
Median Change in Cluster of Differentiation 4 (CD4+) Cell Count From Baseline in TMC125-C229 Feeder Study at Week 192
149.50 x 1000000 cells/mL
Interval -535.0 to 1847.0

SECONDARY outcome

Timeframe: Baseline and Endpoint (ie, the last available time point during the treatment period)

Population: Intent-to-treat population: Participants who received at least 1 dose of study medication were included

Emerging mutations are the mutation which are not present at baseline (last visit of the TMC125 feeder study \[TMC125-C203 (NCT00412646), TMC125-C223 (NCT00081978), TMC125 C211 (NCT00111280) or TMC125-C209 feeder studies\]) and are present at endpoint (last available timepoint during treatment period for each individual participant).

Outcome measures

Outcome measures
Measure
Viral Load More Than or Equal to 50 Copies/mL
n=211 Participants
Viral load more than or equal to 50 copies/mL at TMC125-C229 Baseline
Viral Load Less Than 50 Copies/mL
Viral load less than 50 copies/mL at TMC125-C229 Baseline
Number of Participants With Emerging Mutation (Reverse Transcriptase Mutation)
L100I
8 Participants
Number of Participants With Emerging Mutation (Reverse Transcriptase Mutation)
Y181C
7 Participants
Number of Participants With Emerging Mutation (Reverse Transcriptase Mutation)
A98G
6 Participants
Number of Participants With Emerging Mutation (Reverse Transcriptase Mutation)
V179I
6 Participants
Number of Participants With Emerging Mutation (Reverse Transcriptase Mutation)
K103N
5 Participants
Number of Participants With Emerging Mutation (Reverse Transcriptase Mutation)
H221Y
5 Participants

Adverse Events

Etravirine

Serious events: 46 serious events
Other events: 147 other events
Deaths: 0 deaths

Serious adverse events

Serious adverse events
Measure
Etravirine
n=211 participants at risk
800 mg twice daily (formulation TF035), and after formulation switch, 200 mg twice daily (formulation F060)
Blood and lymphatic system disorders
Febrile neutropenia
0.47%
1/211 • Up to 3 years
Cardiac disorders
Acute coronary syndrome
0.47%
1/211 • Up to 3 years
Cardiac disorders
Acute myocardial infarction
0.47%
1/211 • Up to 3 years
Cardiac disorders
Angina pectoris
0.47%
1/211 • Up to 3 years
Cardiac disorders
Angina unstable
0.47%
1/211 • Up to 3 years
Cardiac disorders
Arrhythmia
0.47%
1/211 • Up to 3 years
Cardiac disorders
Atrial flutter
0.47%
1/211 • Up to 3 years
Cardiac disorders
Cardiogenic shock
0.47%
1/211 • Up to 3 years
Cardiac disorders
Coronary artery disease
0.47%
1/211 • Up to 3 years
Cardiac disorders
Coronary artery occlusion
0.47%
1/211 • Up to 3 years
Cardiac disorders
Myocardial infarction
0.95%
2/211 • Up to 3 years
Cardiac disorders
Myocardial ischaemia
0.47%
1/211 • Up to 3 years
Congenital, familial and genetic disorders
Fanconi syndrome
0.47%
1/211 • Up to 3 years
Endocrine disorders
Adrenal insufficiency
0.95%
2/211 • Up to 3 years
Gastrointestinal disorders
Abdominal distension
0.47%
1/211 • Up to 3 years
Gastrointestinal disorders
Diarrhoea haemorrhagic
0.47%
1/211 • Up to 3 years
Gastrointestinal disorders
Gastritis
0.95%
2/211 • Up to 3 years
Gastrointestinal disorders
Pancreatitis
0.95%
2/211 • Up to 3 years
Gastrointestinal disorders
Upper gastrointestinal haemorrhage
0.47%
1/211 • Up to 3 years
General disorders
Chest discomfort
0.47%
1/211 • Up to 3 years
General disorders
Chills
0.47%
1/211 • Up to 3 years
General disorders
Pyrexia
0.47%
1/211 • Up to 3 years
Hepatobiliary disorders
Cholecystitis
0.47%
1/211 • Up to 3 years
Hepatobiliary disorders
Cholecystitis acute
0.47%
1/211 • Up to 3 years
Infections and infestations
Acute sinusitis
0.47%
1/211 • Up to 3 years
Infections and infestations
Arthritis bacterial
0.47%
1/211 • Up to 3 years
Infections and infestations
Arthritis infective
0.47%
1/211 • Up to 3 years
Infections and infestations
Bacteraemia
0.47%
1/211 • Up to 3 years
Infections and infestations
Bronchitis
0.47%
1/211 • Up to 3 years
Infections and infestations
Cellulitis
1.4%
3/211 • Up to 3 years
Infections and infestations
Gastrointestinal infection
0.47%
1/211 • Up to 3 years
Infections and infestations
Groin abscess
0.47%
1/211 • Up to 3 years
Infections and infestations
Herpes simplex
0.47%
1/211 • Up to 3 years
Infections and infestations
Histoplasmosis disseminated
0.47%
1/211 • Up to 3 years
Infections and infestations
Meningitis aseptic
0.47%
1/211 • Up to 3 years
Infections and infestations
Pneumocystis jiroveCI pneumonia
0.95%
2/211 • Up to 3 years
Infections and infestations
Pneumonia
2.4%
5/211 • Up to 3 years
Infections and infestations
Pneumonia viral
0.47%
1/211 • Up to 3 years
Infections and infestations
Respiratory tract infection
0.47%
1/211 • Up to 3 years
Infections and infestations
Secondary syphilis
0.47%
1/211 • Up to 3 years
Infections and infestations
Sepsis
0.47%
1/211 • Up to 3 years
Infections and infestations
Staphylococcal abscess
0.47%
1/211 • Up to 3 years
Infections and infestations
Subcutaneous abscess
0.47%
1/211 • Up to 3 years
Infections and infestations
Urinary tract infection
0.47%
1/211 • Up to 3 years
Injury, poisoning and procedural complications
Femur fracture
0.47%
1/211 • Up to 3 years
Injury, poisoning and procedural complications
Hip fracture
0.47%
1/211 • Up to 3 years
Injury, poisoning and procedural complications
Injury
0.47%
1/211 • Up to 3 years
Injury, poisoning and procedural complications
Radius fracture
0.47%
1/211 • Up to 3 years
Injury, poisoning and procedural complications
Tibia fracture
0.47%
1/211 • Up to 3 years
Injury, poisoning and procedural complications
Traumatic brain injury
0.47%
1/211 • Up to 3 years
Investigations
Biopsy kidney
0.47%
1/211 • Up to 3 years
Investigations
Biopsy liver
0.47%
1/211 • Up to 3 years
Metabolism and nutrition disorders
Dehydration
0.95%
2/211 • Up to 3 years
Metabolism and nutrition disorders
Diabetes mellitus non-insulin-dependent
0.47%
1/211 • Up to 3 years
Metabolism and nutrition disorders
Metabolic acidosis
0.47%
1/211 • Up to 3 years
Musculoskeletal and connective tissue disorders
Muscle spasms
0.47%
1/211 • Up to 3 years
Musculoskeletal and connective tissue disorders
Musculoskeletal chest pain
0.47%
1/211 • Up to 3 years
Musculoskeletal and connective tissue disorders
Osteoarthritis
0.47%
1/211 • Up to 3 years
Musculoskeletal and connective tissue disorders
Osteonecrosis
0.47%
1/211 • Up to 3 years
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Anal cancer recurrent
0.47%
1/211 • Up to 3 years
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Breast cancer
0.47%
1/211 • Up to 3 years
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Gum neoplasm malignant stage unspecified
0.47%
1/211 • Up to 3 years
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Hepatic neoplasm
0.47%
1/211 • Up to 3 years
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Hepatic neoplasm malignant
0.47%
1/211 • Up to 3 years
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Hodgkin's disease
0.47%
1/211 • Up to 3 years
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Kaposi's sarcoma
0.47%
1/211 • Up to 3 years
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Metastases to liver
0.47%
1/211 • Up to 3 years
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Metastases to peritoneum
0.47%
1/211 • Up to 3 years
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Pancreatic neoplasm
0.47%
1/211 • Up to 3 years
Neoplasms benign, malignant and unspecified (incl cysts and polyps)
Prostate cancer
0.47%
1/211 • Up to 3 years
Nervous system disorders
Chronic inflammatory demyelinating polyradiculoneuropathy
0.47%
1/211 • Up to 3 years
Nervous system disorders
Headache
0.47%
1/211 • Up to 3 years
Renal and urinary disorders
Renal artery occlusion
0.47%
1/211 • Up to 3 years
Renal and urinary disorders
Renal failure acute
0.95%
2/211 • Up to 3 years
Renal and urinary disorders
Renal impairment
0.47%
1/211 • Up to 3 years
Reproductive system and breast disorders
Prostatitis
0.47%
1/211 • Up to 3 years
Respiratory, thoracic and mediastinal disorders
Dyspnoea
0.47%
1/211 • Up to 3 years
Respiratory, thoracic and mediastinal disorders
Pulmonary artery thrombosis
0.47%
1/211 • Up to 3 years
Skin and subcutaneous tissue disorders
Decubitus ulcer
0.47%
1/211 • Up to 3 years
Surgical and medical procedures
Abdominoplasty
0.47%
1/211 • Up to 3 years
Surgical and medical procedures
Hospitalisation
0.47%
1/211 • Up to 3 years
Surgical and medical procedures
Wound treatment
0.47%
1/211 • Up to 3 years
Vascular disorders
Hypertension
0.47%
1/211 • Up to 3 years

Other adverse events

Other adverse events
Measure
Etravirine
n=211 participants at risk
800 mg twice daily (formulation TF035), and after formulation switch, 200 mg twice daily (formulation F060)
Blood and lymphatic system disorders
Lymphadenopathy
10.4%
22/211 • Up to 3 years
Gastrointestinal disorders
Abdominal pain
7.6%
16/211 • Up to 3 years
Gastrointestinal disorders
Diarrhoea
17.5%
37/211 • Up to 3 years
Gastrointestinal disorders
Nausea
8.5%
18/211 • Up to 3 years
Gastrointestinal disorders
Vomiting
5.2%
11/211 • Up to 3 years
General disorders
Fatigue
10.9%
23/211 • Up to 3 years
General disorders
Injection site reaction
7.1%
15/211 • Up to 3 years
General disorders
Pyrexia
7.6%
16/211 • Up to 3 years
Infections and infestations
Bronchitis
7.1%
15/211 • Up to 3 years
Infections and infestations
Nasopharyngitis
10.9%
23/211 • Up to 3 years
Infections and infestations
Sinusitis
11.4%
24/211 • Up to 3 years
Infections and infestations
Upper respiratory tract infection
17.1%
36/211 • Up to 3 years
Musculoskeletal and connective tissue disorders
Arthralgia
10.9%
23/211 • Up to 3 years
Musculoskeletal and connective tissue disorders
Back pain
9.0%
19/211 • Up to 3 years
Musculoskeletal and connective tissue disorders
Myalgia
5.7%
12/211 • Up to 3 years
Musculoskeletal and connective tissue disorders
Pain in extremity
6.2%
13/211 • Up to 3 years
Nervous system disorders
Headache
9.5%
20/211 • Up to 3 years
Psychiatric disorders
Depression
5.2%
11/211 • Up to 3 years
Respiratory, thoracic and mediastinal disorders
Cough
9.5%
20/211 • Up to 3 years
Skin and subcutaneous tissue disorders
Rash
7.6%
16/211 • Up to 3 years
Vascular disorders
Hypertension
5.2%
11/211 • Up to 3 years

Additional Information

Trial Physician

Tibotec Pharmaceuticals

Phone: +32-14-607-767

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place

Restriction type: GT60