Paclitaxel With / Without GW572016 (Lapatinib) As First Line Therapy For Women With Advanced Or Metastatic Breast Cancer

NCT ID: NCT00075270

Last Updated: 2015-05-06

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

580 participants

Study Classification

INTERVENTIONAL

Study Start Date

2004-01-31

Study Completion Date

2012-03-31

Brief Summary

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The purpose of this study is to determine the efficacy and safety of an oral dual tyrosine kinase inhibitor (GW572016) in combination with paclitaxel compared to paclitaxel alone in first line advanced or metastatic breast cancer.

Detailed Description

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Conditions

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Neoplasms, Breast

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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Arm 1

Lapatinib 1500 mg, once daily and Paclitaxel 175 mg/m Intravenously over 3 hours ever 3 weeks

Group Type EXPERIMENTAL

Paclitaxel

Intervention Type DRUG

Active Comparator

GW572016 (Lapatinib)

Intervention Type DRUG

Oral GW572016 Lapatinib

Arm 2

Paclitaxel 175 mg/m Intravenously over 3 hours ever 3 weeks and Placebo

Group Type PLACEBO_COMPARATOR

Paclitaxel

Intervention Type DRUG

Active Comparator

Interventions

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Paclitaxel

Active Comparator

Intervention Type DRUG

GW572016 (Lapatinib)

Oral GW572016 Lapatinib

Intervention Type DRUG

Other Intervention Names

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Paclitaxel

Eligibility Criteria

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Inclusion Criteria

* Signed Informed Consent
* Able to swallow an oral medication
* Cardiac ejection fraction within the institutional range of normal as measured by echocardiogram
* Adequate kidney and liver function
* Adequate bone marrow function
* Tumor tissue available for testing
* Prior adjuvant or neoadjuvant therapy is permitted with an anthracycline or anthracenedione-containing regimen however, subjects must have had cumulative doses of less than 360 mg/m2 of doxorubicin, 720 mg/m2 of epirubicin, or 72 mg/m2 of mitoxantrone
* No Her2/neu overexpression in tumor tissue tested or status unknown if tissue has never been tested

Exclusion Criteria

* Prior treatment regimens for advanced or metastatic breast cancer.
* Pregnant or lactating
* Conditions that would effect the absorption of an oral drug
* Active infection
* Brain metastases
* Treatment with EGFR (Endothelial Growth Factor Receptor) inhibitor.
* Known hypersensitivity to Taxol or excipients of Taxol
* Peripheral neuropathy of Grade 2 or greater is not permitted
* Severe Cardiovascular disease or cardiac disease requiring a device.
* Serious medical or psychiatric disorder that would interfere with the patient's safety or informed consent.
Minimum Eligible Age

18 Years

Eligible Sex

FEMALE

Accepts Healthy Volunteers

No

Sponsors

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GlaxoSmithKline

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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GSK Clinical Trials

Role: STUDY_DIRECTOR

GlaxoSmithKline

Locations

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Tucson, Arizona, United States

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Hot Springs, Arkansas, United States

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Jonesboro, Arkansas, United States

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Fountain Valley, California, United States

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La Jolla, California, United States

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Rancho Mirage, California, United States

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Vallejo, California, United States

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Denver, Colorado, United States

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Boca Raton, Florida, United States

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Orlando, Florida, United States

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Port Saint Lucie, Florida, United States

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West Palm Beach, Florida, United States

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Atlanta, Georgia, United States

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Marietta, Georgia, United States

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Savannah, Georgia, United States

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Savannah, Georgia, United States

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Indianapolis, Indiana, United States

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Kansas City, Kansas, United States

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Metairie, Louisiana, United States

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Baltimore, Maryland, United States

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Glen Burnie, Maryland, United States

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Springfield, Massachusetts, United States

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Duluth, Minnesota, United States

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Robbinsdale, Minnesota, United States

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St Louis, Missouri, United States

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Voorhees Township, New Jersey, United States

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Santa Fe, New Mexico, United States

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Nyack, New York, United States

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Syracuse, New York, United States

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Charlotte, North Carolina, United States

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Greenville, North Carolina, United States

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Fargo, North Dakota, United States

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Canton, Ohio, United States

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Portland, Oregon, United States

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Columbia, South Carolina, United States

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Knoxville, Tennessee, United States

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Knoxville, Tennessee, United States

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Amarillo, Texas, United States

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Fort Worth, Texas, United States

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Houston, Texas, United States

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San Antonio, Texas, United States

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Burlington, Vermont, United States

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Norfolk, Virginia, United States

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Tacoma, Washington, United States

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Milwaukee, Wisconsin, United States

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Buenos Aires, Buenos Aires, Argentina

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Capital Federal, Buenos Aires, Argentina

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Capital Federal, Buenos Aires, Argentina

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Fitzroy, Victoria, Australia

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Malvern, Victoria, Australia

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Wodonga, Victoria, Australia

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Nedlands, Western Australia, Australia

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Vienna, , Austria

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Bruges, , Belgium

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Brussels, , Belgium

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Brussels, , Belgium

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Kortrijk, , Belgium

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Leuven, , Belgium

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Roeselare, , Belgium

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Salvador, Estado de Bahia, Brazil

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Rio de Janeiro, Rio de Janeiro, Brazil

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St. John's, Newfoundland and Labrador, Canada

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Greater Sudbury, Ontario, Canada

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Thunder Bay, Ontario, Canada

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Montreal, Quebec, Canada

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Montreal, Quebec, Canada

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Sherbrooke, Quebec, Canada

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Santiago, Región Metro de Santiago, Chile

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Santiago, Región Metro de Santiago, Chile

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Santiago, Región Metro de Santiago, Chile

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Brno, , Czechia

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Hradec Králové, , Czechia

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Olomouc, , Czechia

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Aalen, Baden-Wurttemberg, Germany

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Stuttgart, Baden-Wurttemberg, Germany

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Ulm, Baden-Wurttemberg, Germany

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Augsburg, Bavaria, Germany

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Bayreuth, Bavaria, Germany

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Coburg, Bavaria, Germany

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Munich, Bavaria, Germany

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Munich, Bavaria, Germany

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Fürstenwalde, Brandenburg, Germany

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Hamburg, City state of Hamburg, Germany

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Hamburg, City state of Hamburg, Germany

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Hamburg, City state of Hamburg, Germany

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Stade, Lower Saxony, Germany

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Herne, North Rhine-Westphalia, Germany

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Ibbenbueren, North Rhine-Westphalia, Germany

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Münster, North Rhine-Westphalia, Germany

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Halle, Saxony-Anhalt, Germany

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Kiel, Schleswig-Holstein, Germany

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Berlin, State of Berlin, Germany

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Berlin, State of Berlin, Germany

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Berlin, State of Berlin, Germany

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Berlin, State of Berlin, Germany

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Jena, Thuringia, Germany

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Budapest, , Hungary

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Nyíregyháza, , Hungary

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Szombathely, , Hungary

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Zalaegerszeg-Pózva, , Hungary

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Benevento, Campania, Italy

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Napoli, Campania, Italy

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Forlì, Emilia-Romagna, Italy

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Parma, Emilia-Romagna, Italy

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Ravenna, Emilia-Romagna, Italy

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Rimini, Emilia-Romagna, Italy

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Rome, Lazio, Italy

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Rome, Lazio, Italy

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Pietra Ligure (SV), Liguria, Italy

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Bergamo, Lombardy, Italy

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Pavia, Lombardy, Italy

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Candiolo (TO), Piedmont, Italy

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Turin, Piedmont, Italy

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Sassari, Sardinia, Italy

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Prato (PO), Tuscany, Italy

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Perugia, Umbria, Italy

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Daugavpils, , Latvia

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Liepāja, , Latvia

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Riga, , Latvia

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Riga, , Latvia

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Colima, Colima, Mexico

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Durango, Durango, Mexico

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Acapulco de Juárez, Guerrero, Mexico

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Guadalajara, Jalisco, Mexico

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Amersfoort, , Netherlands

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Leiden, , Netherlands

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Nieuwegein, , Netherlands

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Utrecht, , Netherlands

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Utrecht, , Netherlands

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Auckland, , New Zealand

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Christchurch, , New Zealand

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Lahore, , Pakistan

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Lahore, , Pakistan

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Lima, Lima Province, Peru

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Callao, , Peru

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Krakow, , Poland

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Olsztyn, , Poland

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Olsztyn, , Poland

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Poznan, , Poland

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Warsaw, , Poland

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Wroclaw, , Poland

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Moscow, , Russia

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Moscow, , Russia

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Moscow, , Russia

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Moscow, , Russia

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Moscow, , Russia

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Moscow Region, , Russia

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Saint Petersburg, , Russia

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Saint Petersburg, , Russia

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Banská Bystrica, , Slovakia

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Bratislava, , Slovakia

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Košice, , Slovakia

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Poprad, , Slovakia

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Parktown, Gauteng, South Africa

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Capital Park, , South Africa

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Overport, , South Africa

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Parow, , South Africa

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Port Elizabeth, , South Africa

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Gyeonggi-do, , South Korea

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Seoul, , South Korea

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Alcorcón/Madrid, , Spain

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Baracaldo/Vizcaya, , Spain

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Cáceres, , Spain

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Cuidad Real, , Spain

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Jaén, , Spain

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La Laguna (Santa Cruz de Tenerife), , Spain

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Las Palmas de Gran Canaria, , Spain

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Madrid, , Spain

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Móstoles/Madrid, , Spain

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Palma de Mallorca, , Spain

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Pontevedra, , Spain

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San Sebastián, , Spain

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Santa Cruz de Tenerife, , Spain

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Zaragoza, , Spain

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Zaragoza, , Spain

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Istanbul, , Turkey (Türkiye)

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Istanbul, , Turkey (Türkiye)

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Countries

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United States Argentina Australia Austria Belgium Brazil Canada Chile Czechia Germany Hungary Italy Latvia Mexico Netherlands New Zealand Pakistan Peru Poland Russia Slovakia South Africa South Korea Spain Turkey (Türkiye)

References

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Tenori L, Oakman C, Claudino WM, Bernini P, Cappadona S, Nepi S, Biganzoli L, Arbushites MC, Luchinat C, Bertini I, Di Leo A. Exploration of serum metabolomic profiles and outcomes in women with metastatic breast cancer: a pilot study. Mol Oncol. 2012 Aug;6(4):437-44. doi: 10.1016/j.molonc.2012.05.003. Epub 2012 Jun 1.

Reference Type BACKGROUND
PMID: 22687601 (View on PubMed)

Finn RS, Press MF, Dering J, Arbushites M, Koehler M, Oliva C, Williams LS, Di Leo A. Estrogen receptor, progesterone receptor, human epidermal growth factor receptor 2 (HER2), and epidermal growth factor receptor expression and benefit from lapatinib in a randomized trial of paclitaxel with lapatinib or placebo as first-line treatment in HER2-negative or unknown metastatic breast cancer. J Clin Oncol. 2009 Aug 20;27(24):3908-15. doi: 10.1200/JCO.2008.18.1925. Epub 2009 Jul 20.

Reference Type BACKGROUND
PMID: 19620495 (View on PubMed)

Sherrill B, Di Leo A, Amonkar MM, Wu Y, Zvirbule Z, Aziz Z, Bines J, Gomez HL. Quality-of-life and quality-adjusted survival (Q-TWiST) in patients receiving lapatinib in combination with paclitaxel as first-line treatment for metastatic breast cancer. Curr Med Res Opin. 2010 Apr;26(4):767-75. doi: 10.1185/03007991003590860.

Reference Type DERIVED
PMID: 20095796 (View on PubMed)

Other Identifiers

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EGF30001

Identifier Type: -

Identifier Source: org_study_id

NCT00085046

Identifier Type: -

Identifier Source: nct_alias

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